Lormetazepam

Lormetazepam

SCHEMBL43267

CN1C(=O)C(O)N=C(c2ccccc2Cl)c2cc(Cl)ccc21

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
OPRK1 P41145 3/20 1.00
PDE4D Q08499 2/20 1.00
CHRM2 P08172 1/20 1.00
ADRA2A P08913 1/20 1.00
LMNA P02545 3/20 0.76
PDE3A Q14432 1/20 0.76
PGR P06401 1/20 0.60
HTR2B P41595 1/20 0.50
GABRA1 P14867 3/20 0.48
GABRA5 P31644 3/20 0.48
GABRA2 P47869 3/20 0.48
GABRB2 P47870 3/20 0.48
GABRP O00591 2/20 0.48
GABRD O14764 2/20 0.48
GABRB1 P18505 2/20 0.48
GABRG2 P18507 2/20 0.48
GABRB3 P28472 2/20 0.48
GABRA3 P34903 2/20 0.48
GABRA4 P48169 2/20 0.48
GABRE P78334 2/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Lormetazepam SCHEMBL29565149 1.00 OPRK1 (1.00) OPRK1PDE4DCHRM2ADRA2ALMNA
Lormetazepam SCHEMBL29484438 1.00 OPRK1 (1.00) OPRK1PDE4DCHRM2ADRA2ALMNA
(S)-Lormetazepam SCHEMBL43268 1.00 OPRK1 (1.00) OPRK1PDE4DCHRM2ADRA2ALMNA
Lormetazepam SCHEMBL1758605 0.94 OPRK1 (0.89) OPRK1PDE4DCHRM2ADRA2ALMNA
Lormetazepam SCHEMBL21295409 0.92 OPRK1 (0.85) OPRK1PDE4DCHRM2ADRA2ALMNA
Flutemazepam SCHEMBL1006405 0.88 OPRK1 (0.79) OPRK1PDE4DCHRM2ADRA2ALMNA
Flutemazepam SCHEMBL1006406 0.88 OPRK1 (0.79) OPRK1PDE4DCHRM2ADRA2ALMNA
Temazepam SCHEMBL5503177 0.86 OPRK1 (1.00) OPRK1PDE4DCHRM2ADRA2ALMNA
Temazepam SCHEMBL29463 0.86 OPRK1 (1.00) OPRK1PDE4DCHRM2ADRA2ALMNA
SCHEMBL6944910 0.86 OPRK1 (0.76) OPRK1PDE4DCHRM2ADRA2ALMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 6755 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20260115161-A1 2-HYDROXY-OCTADECENE-9-CIS-OATE FOR USE IN THE TREATMENT OF ONCOLOGICAL PATHOLOGIES AND NEUROPATHIC PAIN LAMINAR PHARMACEUTICALS S A (ES) 2026-04-30 US claimed
EP-4719552-A1 INDUCTION OF GENERAL ANESTHESIA IN ADULTS UNDERGOING ELECTIVE SURGERY Xizang Haisco Pharmaceutical Co., Ltd. (CN) 2026-04-08 EP claimed
US-20260076953-A1 METHODS OF DIAGNOSING AND TREATING ADHD IN BIOMARKER POSITIVE SUBJECTS THE CHILDREN'S HOSPITAL OF PHILADELPHIA (US) 2026-03-19 US claimed
EP-3507371-B1 COMPOSITIONS FOR TREATING DISEASES AND DISORDERS OF THE NERVOUS SYSTEM UNIV RUTGERS (US) 2026-01-28 EP claimed
EP-4663187-A1 2-HYDROXY-OCTADECENE-9-CIS-OATE FOR USE IN THE TREATMENT OF ONCOLOGICAL PATHOLOGIES AND NEUROPATHIC PAIN Laminar Pharmaceuticals, S.A. (ES) 2025-12-17 EP claimed
US-20250375421-A1 METHODS OF USING DMT SHULMAN WILLIAM (US) 2025-12-11 US claimed
US-12396981-B2 Methods of using DMT SHULMAN WILLIAM (US) 2025-08-26 US claimed
US-20250120962-A1 NONSELECTIVE METABOTROPIC GLUTAMATE RECEPTOR ACTIVATORS FOR TREATMENT OF ATTENTION DEFICIT DISORDER AND 22Q SYNDROME THE CHILDREN'S HOSPITAL OF PHILADELPHIA (US) 2025-04-17 US claimed
EP-4023222-B1 NONSELECTIVE METABOTROPIC GLUTAMATE RECEPTOR ACTIVATOR FOR TREATMENT OF 22Q SYNDROME CHILDRENS HOSPITAL PHILADELPHIA (US) 2024-12-18 EP claimed
WO-2024251110-A1 INDUCTION OF GENERAL ANESTHESIA IN ADULTS UNDERGOING ELECTIVE SURGERY XIZANG HAISCO PHARMACEUTICAL CO., LTD. (CN) 2024-12-12 WO claimed
EP-0682943-A1 Oil-in-water emulsion containing lorazepam or lormetazepam GESELLSCHAFT FÜR MEDIZINISCHE FORSCHUNG UND WEITERBILDUNG e.V. GMF (DE) 1995-11-22 EP claimed
EP-0584285-A1 IMPROVEMENTS IN BENZODIAZEPINE TREATMENT BY CHOLINESTERASE INHIBITORS Snorrason, Ernir (IS) 1994-03-02 EP claimed
US-5288497-A Compositions of oral dissolvable medicaments THE UNIVERSITY OF UTAH (US) 1994-02-22 US claimed
US-5288498-A Compositions of oral nondissolvable matrixes for transmucosal administration of medicaments UNIVERSITY OF UTAH RESEARCH FOUNDATION (US) 1994-02-22 US claimed
EP-0579435-A1 Cyclodextrin complexation CYCLOPS h.f. (IS) 1994-01-19 EP claimed
US-5248678-A Administering adenosine receptor antagonist and a GABA antagonist FRACTAL LABORATORIES, INC. (US) 1993-09-28 US claimed
WO-1992020328-A2 IMPROVEMENTS IN BENZODIAZEPINE TREATMENT BY CHOLINESTERASE INHIBITORS SNORRASON ERNIR (IS) 1992-11-26 WO claimed
EP-0515301-A2 Improvements in benzodiazepine treatment by cholinesterterase inhibitors Snorrason, Ernir (IS) 1992-11-25 EP claimed
US-4721709-A Novel pharmaceutical compositions containing hydrophobic practically water-insoluble drugs adsorbed on pharmaceutical excipients as carrier; process for their preparation and the use of said compositions PYARE SETH (CH) 1988-01-26 US claimed
US-4065451-A CNS DEPRESSANTS AMERICAN HOME PRODUCTS (US) 1977-12-27 US claimed