Temazepam

Temazepam

SCHEMBL29463

CN1C(=O)C(O)N=C(c2ccccc2)c2cc(Cl)ccc21

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

GABRA1GABRA2GABRA3GABRA4GABRA5GABRA6GABRB1GABRB2GABRB3GABRDGABREGABRG1GABRG2GABRG3GABRPGABRQ

The experimentally established mechanism targets of Temazepam. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GABRP known ✓ O00591 2/20 0.59
GABRD known ✓ O14764 2/20 0.59
GABRA1 known ✓ P14867 2/20 0.59
GABRB1 known ✓ P18505 2/20 0.59
GABRG2 known ✓ P18507 2/20 0.59
GABRB3 known ✓ P28472 2/20 0.59
GABRA5 known ✓ P31644 2/20 0.59
GABRA3 known ✓ P34903 2/20 0.59
GABRA2 known ✓ P47869 2/20 0.59
GABRB2 known ✓ P47870 2/20 0.59
GABRA4 known ✓ P48169 2/20 0.59
GABRE known ✓ P78334 2/20 0.59
GABRA6 known ✓ Q16445 2/20 0.59
GABRG1 known ✓ Q8N1C3 2/20 0.59
GABRG3 known ✓ Q99928 2/20 0.59
GABRQ known ✓ Q9UN88 2/20 0.59
OPRK1 P41145 3/20 1.00
LMNA P02545 2/20 1.00
PDE3A Q14432 1/20 1.00
PDE4D Q08499 2/20 0.76

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Temazepam SCHEMBL29398512 1.00 OPRK1 (1.00) OPRK1LMNAPDE3APDE4DCHRM2
Temazepam SCHEMBL5503177 1.00 OPRK1 (1.00) OPRK1LMNAPDE3APDE4DCHRM2
Temazepam SCHEMBL81963 1.00 OPRK1 (1.00) OPRK1LMNAPDE3APDE4DCHRM2
Temazepam SCHEMBL29464 1.00 OPRK1 (1.00) OPRK1LMNAPDE3APDE4DCHRM2
Temazepam SCHEMBL16922195 1.00 OPRK1 (1.00) OPRK1LMNAPDE3APDE4DCHRM2
Temazepam SCHEMBL10480110 0.99 OPRK1 (0.98) OPRK1LMNAPDE3APDE4DCHRM2
Lormetazepam SCHEMBL1758605 0.93 OPRK1 (0.89) OPRK1LMNAPDE3APDE4DCHRM2
Temazepam SCHEMBL23038565 0.91 OPRK1 (0.83) OPRK1LMNAPDE3APDE4DCHRM2
Temazepam SCHEMBL8140373 0.91 OPRK1 (0.83) OPRK1LMNAPDE3APDE4DCHRM2
Temazepam SCHEMBL7036032 0.90 OPRK1 (0.82) OPRK1LMNAPDE3APDE4DCHRM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 28171 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12624037-B2 Method of treating agitation, aggressive behavior, and impulse control disorder INTRA-CELLULAR THERAPIES, INC. (US) 2026-05-12 US claimed
US-12624036-B2 Method of treating post-traumatic stress disorder INTRA-CELLULAR THERAPIES, INC. (US) 2026-05-12 US claimed
WO-2026090360-A1 FUSED PYRIMIDINE COMPOUNDS FOR TREATMENT OF TINNITUS, HEARING LOSS, AND MENIERE'S DISEASE OVID THERAPEUTICS INC. (US) 2026-04-30 WO claimed
US-20260108529-A1 FUSED AMINO PYRIMIDINE COMPOUNDS FOR TREATMENT OF TINNITUS, ACUTE SENSORINEURAL HEARING LOSS, AGE-RELATED HEARING LOSS, AND MENIERE'S DISEASE OVID THERAPEUTICS INC (US) 2026-04-23 US claimed
US-12594388-B2 Device to deliver a predetermined amount of a substance to a natural orifice of the body APTARGROUP, INC. (US) 2026-04-07 US claimed
US-20260076953-A1 METHODS OF DIAGNOSING AND TREATING ADHD IN BIOMARKER POSITIVE SUBJECTS THE CHILDREN'S HOSPITAL OF PHILADELPHIA (US) 2026-03-19 US claimed
US-20260027337-A1 TRANSDERMAL DRUG DELIVERY DEVICES AND METHODS MORNINGSIDE VENTURE INVESTMENTS LTD (MC) 2026-01-29 US claimed
EP-3507371-B1 COMPOSITIONS FOR TREATING DISEASES AND DISORDERS OF THE NERVOUS SYSTEM UNIV RUTGERS (US) 2026-01-28 EP claimed
EP-4680203-A1 COMPOSITIONS FOR SUSTAINED RELEASE OF POORLY SOLUBLE ACTIVE INGREDIENTS Prolevi Bio AB (SE) 2026-01-21 EP claimed
US-12515030-B2 Transdermal drug delivery devices and methods MORNINGSIDE VENTURE INVESTMENTS LIMITED (MC) 2026-01-06 US claimed
EP-0098113-A1 A combination of beta-adrenoceptor antagonists and anxiolytic agents AYERST, MCKENNA AND HARRISON INC. (CA) 1984-01-11 EP claimed
WO-1983003968-A1 BRAIN-SPECIFIC DRUG DELIVERY UNIVERSITY OF FLORIDA (US) 1983-11-24 WO claimed
EP-0092179-A1 Embedding unit of paving stones for producing soil covers, and process for producing the paving units and soil covers Heinrich-Ludwig Wahrendorf oHG (DE) 1983-10-26 EP claimed
EP-0081194-A1 Bituminous pavement repair method Schölkopf, Walter (DE) 1983-06-15 EP claimed
EP-0072491-A1 Brake for rolling containers Lermer GmbH (DE) 1983-02-23 EP claimed
US-4369172-A Prolonged release therapeutic compositions based on hydroxypropylmethylcellulose FOREST LABORATORIES INC. (US) 1983-01-18 US claimed
EP-0060044-A1 Fluidised bed combustion EMS THERMPLANT LIMITED (GB) 1982-09-15 EP claimed
US-4316897-A TRANQUILIZERS HOFFMANN-LA ROCHE INC. (US) 1982-02-23 US claimed
EP-0025546-A2 Therapeutical use of tranquillizing benzodiazepine derivatives and mixtures containing them F. HOFFMANN-LA ROCHE & CO. Aktiengesellschaft (CH) 1981-03-25 EP claimed
US-4065451-A CNS DEPRESSANTS AMERICAN HOME PRODUCTS (US) 1977-12-27 US claimed