SCHEMBL43292

SCHEMBL43292

N[C@@H](Cc1cccs1)C(=O)O

nearest known ligand 0.70

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CYP2C19 P33261 1/20 0.70
CTSC P53634 12/20 0.61
SLC1A3 P43003 1/20 0.55
SLC1A2 P43004 1/20 0.55
SLC1A1 P43005 1/20 0.55
ALPI P09923 1/20 0.53
PKM P14618 1/20 0.53
PTGS1 P23219 1/20 0.53
XIAP P98170 1/20 0.53
SLC7A5 Q01650 1/20 0.53
RAB9A P51151 1/20 0.51
POLB P06746 1/20 0.47
CTSL P07711 1/20 0.47
CTSS P25774 1/20 0.47
DPP4 P27487 1/20 0.47
DPP8 Q6V1X1 1/20 0.47
DPP9 Q86TI2 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL43293 1.00 CYP2C19 (0.70) CYP2C19CTSCSLC1A3SLC1A2SLC1A1
SCHEMBL288244 1.00 CYP2C19 (0.70) CYP2C19CTSCSLC1A3SLC1A2SLC1A1
Hydrochloric Acid SCHEMBL7382497 0.98 CYP2C19 (0.68) CYP2C19CTSCSLC1A3SLC1A2SLC1A1
Hydrochloric Acid SCHEMBL7382495 0.98 CYP2C19 (0.68) CYP2C19CTSCSLC1A3SLC1A2SLC1A1
Glycine SCHEMBL8101008 0.93 CYP2C19 (0.62) CYP2C19CTSCSLC1A3SLC1A2SLC1A1
SCHEMBL5236901 0.89 CYP2C19 (0.57) CYP2C19CTSCSLC1A3SLC1A2SLC1A1
SCHEMBL5236908 0.89 CYP2C19 (0.57) CYP2C19CTSCSLC1A3SLC1A2SLC1A1
SCHEMBL7252652 0.87 CYP2C19 (0.54) CYP2C19CTSCSLC1A3SLC1A2SLC1A1
SCHEMBL7252654 0.87 CYP2C19 (0.54) CYP2C19CTSCSLC1A3SLC1A2SLC1A1
Isoleucine SCHEMBL8483685 0.85 CYP2C19 (0.53) CYP2C19CTSCSLC1A3SLC1A2SLC1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 7221 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20260085092-A1 MELANOCORTIN RECEPTOR LIGANDS IPSEN PHARMA SAS (FR) 2026-03-26 US claimed
EP-4711004-A2 METHOD OF TREATING MELANOCORTIN-4 RECEPTOR PATHWAY-ASSOCIATED DISORDERS Rhythm Pharmaceuticals, Inc. (US) 2026-03-18 EP claimed
US-12521455-B2 Kisspeptin receptor (KISS1R) targeted therapeutics and uses thereof RADIONETICS ONCOLOGY, INC. (US) 2026-01-13 US claimed
US-20260001915-A1 METHODS FOR TREATING OBESITY WITH AN MC4R AGONIST RHYTHM PHARMACEUTICALS INC (US) 2026-01-01 US claimed
EP-4633656-A1 STAPLED PEPTIDES AND METHODS THEREOF Parabilis Medicines, Inc. (US) 2025-10-22 EP claimed
EP-4633657-A1 STAPLED PEPTIDES AND METHODS THEREOF Parabilis Medicines, Inc. (US) 2025-10-22 EP claimed
WO-2025217074-A1 KISSPEPTIN RECEPTOR (KISS1R) TARGETED THERAPEUTICS AND USES THEREOF RADIONETICS ONCOLOGY, INC. (US) 2025-10-16 WO claimed
US-20250295792-A1 POLYETHYLENE GLYCOL-MODIFIED FORM OF KININ OR DERIVATIVE THEREOF AND PHARMACEUTICAL USE THEREOF ZONHON BIOPHARMA INSTITUTE, INC. (CN) 2025-09-25 US claimed
US-20250195606-A1 METHOD OF TREATING MELANOCORTIN-4 RECEPTOR PATHWAY-ASSOCIATED DISORDERS CHARITÉ - UNIVERSITÄTSMEDIZIN BERLIN (DE) 2025-06-19 US claimed
CN-120152725-A Methods of treating obesity using MC4R agonists 节奏制药公司 2025-06-13 CN claimed
US-4693993-A ANTIINFLAMMATORY VAVREK, RAYMOND J. 1987-09-15 US claimed
US-4690936-A AMINO ACIDS, THIOESTER LINKAGE; ANGIOTENSIN INHIBITORS UNIVERSITY OF MIAMI (US) 1987-09-01 US claimed
EP-0230242-A2 Substituted derivatives of 4-amino-3-hydroxy-butyric acid, process for their production, medicines containing them, and their use HOECHST AKTIENGESELLSCHAFT (DE) 1987-07-29 EP claimed
EP-0225386-A1 BRADYKININ ANTAGONIST PEPTIDES NOVA TECHNOLOGY LIMITED PARTNERSHIP (US) 1987-06-16 EP claimed
WO-1986007263-A1 BRADYKININ ANTAGONIST PEPTIDES STEWART JOHN M 1986-12-18 WO claimed
US-4493828-A Use of thyrotropin releasing hormone and related peptides as poultry growth promotants MERCK & CO., INC. (US) 1985-01-15 US claimed
EP-0036713-B1 ANGIOTENSIN CONVERTING ENZYME INHIBITORS UNIVERSITY OF MIAMI (US) 1984-01-18 EP claimed
US-4407952-A OF GENETICALLY ENGINEERED ESCHERICHIA AJINOMOTO COMPANY INCORPORATED (JP) 1983-10-04 US claimed
US-4328134-A Anorexigenic peptides ADMINISTRATORS OF THE TULANE UNIVERSITY EDUCATIONAL FUND, THE, A CORP. OF LA 1982-05-04 US claimed
EP-0036713-A2 Angiotensin converting enzyme inhibitors UNIVERSITY OF MIAMI (US) 1981-09-30 EP claimed