SCHEMBL43293

SCHEMBL43293

NC(Cc1cccs1)C(=O)O

nearest known ligand 0.70

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CYP2C19 P33261 1/20 0.70
CTSC P53634 12/20 0.61
SLC1A3 P43003 1/20 0.55
SLC1A2 P43004 1/20 0.55
SLC1A1 P43005 1/20 0.55
ALPI P09923 1/20 0.53
PKM P14618 1/20 0.53
PTGS1 P23219 1/20 0.53
XIAP P98170 1/20 0.53
SLC7A5 Q01650 1/20 0.53
RAB9A P51151 1/20 0.51
POLB P06746 1/20 0.47
CTSL P07711 1/20 0.47
CTSS P25774 1/20 0.47
DPP4 P27487 1/20 0.47
DPP8 Q6V1X1 1/20 0.47
DPP9 Q86TI2 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL43292 1.00 CYP2C19 (0.70) CYP2C19CTSCSLC1A3SLC1A2SLC1A1
SCHEMBL288244 1.00 CYP2C19 (0.70) CYP2C19CTSCSLC1A3SLC1A2SLC1A1
Hydrochloric Acid SCHEMBL7382497 0.98 CYP2C19 (0.68) CYP2C19CTSCSLC1A3SLC1A2SLC1A1
Hydrochloric Acid SCHEMBL7382495 0.98 CYP2C19 (0.68) CYP2C19CTSCSLC1A3SLC1A2SLC1A1
Glycine SCHEMBL8101008 0.93 CYP2C19 (0.62) CYP2C19CTSCSLC1A3SLC1A2SLC1A1
SCHEMBL5236901 0.89 CYP2C19 (0.57) CYP2C19CTSCSLC1A3SLC1A2SLC1A1
SCHEMBL5236908 0.89 CYP2C19 (0.57) CYP2C19CTSCSLC1A3SLC1A2SLC1A1
SCHEMBL7252652 0.87 CYP2C19 (0.54) CYP2C19CTSCSLC1A3SLC1A2SLC1A1
SCHEMBL7252654 0.87 CYP2C19 (0.54) CYP2C19CTSCSLC1A3SLC1A2SLC1A1
Isoleucine SCHEMBL8483685 0.85 CYP2C19 (0.53) CYP2C19CTSCSLC1A3SLC1A2SLC1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 5172 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12521455-B2 Kisspeptin receptor (KISS1R) targeted therapeutics and uses thereof RADIONETICS ONCOLOGY, INC. (US) 2026-01-13 US claimed
WO-2025217074-A1 KISSPEPTIN RECEPTOR (KISS1R) TARGETED THERAPEUTICS AND USES THEREOF RADIONETICS ONCOLOGY, INC. (US) 2025-10-16 WO claimed
US-20250295792-A1 POLYETHYLENE GLYCOL-MODIFIED FORM OF KININ OR DERIVATIVE THEREOF AND PHARMACEUTICAL USE THEREOF ZONHON BIOPHARMA INSTITUTE, INC. (CN) 2025-09-25 US claimed
US-20250129127-A1 Systems for Amplification of AAV Rep and Cap Proteins SHAPE THERAPEUTICS INC. 2025-04-24 US claimed
US-20240366812-A1 Radiolabeled GRPR-Antagonists for Diagnostic Imaging and Treatment of GRPR-Positive Cancer ADVANCED ACCELERATOR APPLICATIONS INTERNATIONAL SA (CH) 2024-11-07 US claimed
US-20240197896-A1 SYNTHETIC PEPTIDE SHUTTLE AGENT BIOCONJUGATES FOR INTRACELLULAR CARGO DELIVERY FELDAN BIO INC. (CA) 2024-06-20 US claimed
CN-117750978-A Synthetic peptide shuttle bioconjugates for intracellular cargo delivery 费尔丹生物公司 2024-03-22 CN claimed
EP-4313159-A1 SYNTHETIC PEPTIDE SHUTTLE AGENT BIOCONJUGATES FOR INTRACELLULAR CARGO DELIVERY Feldan Bio Inc. (CA) 2024-02-07 EP claimed
US-20230399661-A1 SHUTTLE AGENT PEPTIDES OF MINIMAL LENGTH AND VARIANTS THEREOF ADAPTED FOR TRANSDUCTION OF CAS9-RNP AND OTHER NUCLEOPROTEIN CARGOS FELDAN BIO INC. (CA) 2023-12-14 US claimed
US-20230383291-A1 PEPTIDE-BASED TRANSDUCTION OF NON-ANIONIC POLYNUCLEOTIDE ANALOGS FOR GENE EXPRESSION MODULATION FELDAN BIO INC. (CA) 2023-11-30 US claimed
CN-1035286-A The amino acid derivative of renin-inhibiting HOECHST AG (DE) 1989-09-06 CN claimed
US-4855286-A HYPOTENSIVE AGENTS HOECHST AKTIENGESELLSCHAFT (DE) 1989-08-08 US claimed
EP-0320785-A2 Peptides influencing the activity of the hypophysis of mammalians HOECHST AKTIENGESELLSCHAFT (DE) 1989-06-21 EP claimed
US-4693993-A ANTIINFLAMMATORY VAVREK, RAYMOND J. 1987-09-15 US claimed
US-4690936-A AMINO ACIDS, THIOESTER LINKAGE; ANGIOTENSIN INHIBITORS UNIVERSITY OF MIAMI (US) 1987-09-01 US claimed
EP-0225386-A1 BRADYKININ ANTAGONIST PEPTIDES NOVA TECHNOLOGY LIMITED PARTNERSHIP (US) 1987-06-16 EP claimed
WO-1986007263-A1 BRADYKININ ANTAGONIST PEPTIDES STEWART JOHN M 1986-12-18 WO claimed
EP-0036713-B1 ANGIOTENSIN CONVERTING ENZYME INHIBITORS UNIVERSITY OF MIAMI (US) 1984-01-18 EP claimed
US-4407952-A OF GENETICALLY ENGINEERED ESCHERICHIA AJINOMOTO COMPANY INCORPORATED (JP) 1983-10-04 US claimed
EP-0036713-A2 Angiotensin converting enzyme inhibitors UNIVERSITY OF MIAMI (US) 1981-09-30 EP claimed