SCHEMBL4330968

SCHEMBL4330968

FC(F)(F)c1ccc(COc2cc(-c3ccc(C4CC[CH]CC4)cc3)[nH]n2)cc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PRMT5 O14744 1/20 0.44
HTR2C P28335 3/20 0.38
MRGPRX4 Q96LA9 1/20 0.37
MAOB P27338 3/20 0.36
F10 P00742 1/20 0.36
FEN1 P39748 2/20 0.35
P2RY14 Q15391 1/20 0.35
SLC6A4 P31645 2/20 0.34
RXRA P19793 1/20 0.34
RXRB P28702 1/20 0.34
RXRG P48443 1/20 0.34
TNIK Q9UKE5 1/20 0.34
MAP4K3 Q8IVH8 1/20 0.34
KDM1A O60341 1/20 0.34
MAOA P21397 1/20 0.34
PTPN2 P17706 1/20 0.34
PTPN1 P18031 1/20 0.34
PTPN6 P29350 1/20 0.34
DGAT1 O75907 1/20 0.34
SOAT1 P35610 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4936610 0.84 DGAT1 (0.54) RXRARXRBRXRGPTPN2PTPN1
SCHEMBL4475129 0.81 SLC6A4 (0.39) MRGPRX4MAOBFEN1SLC6A4KDM1A
SCHEMBL4480678 0.81 SLC6A4 (0.40) HTR2CSLC6A4HTR2B
SCHEMBL4491043 0.78 S1PR1 (0.37) HTR2CFEN1SLC6A4GLP1RALOX5AP
SCHEMBL4493691 0.74 IGF1R (0.36) SLC6A4
SCHEMBL4065138 0.71 HTR2C (0.63) HTR2CMAOBKDM1A
SCHEMBL4474532 0.70 CHEK1 (0.37) TNIK
SCHEMBL4487832 0.70 DGAT1 (0.45) DGAT1SOAT1
SCHEMBL14813186 0.66 DGAT1 (0.45) HTR2CSLC6A4DGAT1SOAT1HTR2B
SCHEMBL4920803 0.66 CBFB (0.46) MAOBDGAT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2117526-A2 INHIBITORS OF DIACYLGLYCEROL O-ACYLTRANSFERASE TYPE 1 ENZYME Abbott Laboratories (US) 2009-11-18 EP claimed
WO-2008067257-A2 INHIBITORS OF DIACYLGLYCEROL O-ACYLTRANSFERASE TYPE 1 ENZYME ABBOTT LABORATORIES (US) 2008-06-05 WO claimed
EP-2117526-A2 INHIBITORS OF DIACYLGLYCEROL O-ACYLTRANSFERASE TYPE 1 ENZYME Abbott Laboratories (US) 2009-11-18 EP disclosed
WO-2008067257-A2 INHIBITORS OF DIACYLGLYCEROL O-ACYLTRANSFERASE TYPE 1 ENZYME ABBOTT LABORATORIES (US) 2008-06-05 WO disclosed