SCHEMBL4332819

SCHEMBL4332819

Cc1nc2cc(O)c(-c3nnc(S)n3-c3ccc(C(=O)O)c4ccccc34)cc2[nH]1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DHODH Q02127 8/20 0.38
HSP90AA1 P07900 2/20 0.37
ESR2 Q92731 1/20 0.37
TDP1 Q9NUW8 1/20 0.37
POLB P06746 2/20 0.36
RAB9A P51151 2/20 0.36
ALDH1A1 P00352 2/20 0.36
HPGD P15428 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
MEN1 O00255 1/20 0.32
NPC1 O15118 1/20 0.32
KMT2A Q03164 1/20 0.32
PARP1 P09874 1/20 0.32
TNKS2 Q9H2K2 1/20 0.32
FGFR1 P11362 2/20 0.32
FGFR2 P21802 2/20 0.32
FGFR3 P22607 2/20 0.32
PRKAG1 P54619 1/20 0.32
PRKAA2 P54646 1/20 0.32
PRKAA1 Q13131 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1304644 0.96 DHODH (0.38) DHODHHSP90AA1ESR2TDP1POLB
SCHEMBL14342533 0.85 ALDH1A1 (0.30) POLBRAB9AALDH1A1HPGDSMN1; SMN2
SCHEMBL931684 0.79 TSHR (0.39) HSP90AA1ESR2TDP1POLBRAB9A
SCHEMBL8930899 0.72 MCL1 (0.43) HSP90AA1ALDH1A1HPGDMEN1KMT2A
SCHEMBL931576 0.69 PDK2 (0.37) HSP90AA1ESR2MEN1KMT2A
SCHEMBL12832347 0.69 MCL1 (0.37) HSP90AA1ALDH1A1HPGDMEN1KMT2A
SCHEMBL12047056 0.67 TUBB4A (0.33)
SCHEMBL12832577 0.67 GSK3B (0.31) SMN1; SMN2MEN1KMT2A
SCHEMBL13099831 0.66 HSP90AA1 (0.35) HSP90AA1RAB9ASMN1; SMN2MEN1NPC1
SCHEMBL931360 0.66 ALDH1A1 (0.41) HSP90AA1TDP1POLBRAB9AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2035396-A2 TRIAZOLE COMPOUNDS THAT MODULATE HSP90 ACTIVITY Synta Pharmaceuticals Corporation (US) 2009-03-18 EP claimed
WO-2007139967-A2 TRIAZOLE COMPOUNDS THAT MODULATE HSP90 ACTIVITY SYNTA PHARMACEUTICALS CORP. (US) 2007-12-06 WO claimed