SCHEMBL4333138

SCHEMBL4333138

O=C1NCC=Nc2nc3cccnc3cc21

nearest known ligand 0.33

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.33
PARP10 Q53GL7 1/20 0.33
PARP11 Q9NR21 1/20 0.33
PIM1 P11309 5/20 0.32
PIM2 Q9P1W9 4/20 0.32
CSNK2A1 P68400 2/20 0.32
DYRK1A Q13627 2/20 0.32
CLK4 Q9HAZ1 2/20 0.32
STK17A Q9UEE5 2/20 0.32
MAPKAPK2 P49137 2/20 0.32
PLK4 O00444 1/20 0.32
DAPK3 O43293 1/20 0.32
DYRK3 O43781 1/20 0.32
PRKD3 O94806 1/20 0.32
MAP4K4 O95819 1/20 0.32
CHEK2 O96017 1/20 0.32
CDK1 P06493 1/20 0.32
RPS6KB1 P23443 1/20 0.32
MAPK1 P28482 1/20 0.32
MAPK8 P45983 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2419928 0.82 NPC1 (0.41) ALDH1A1PARP10PARP11PIM1PIM2
SCHEMBL26512083 0.77 TDP2 (0.38) ALDH1A1PARP10PARP11MEN1KMT2A
SCHEMBL2427753 0.74 RAB9A (0.37) ALDH1A1MEN1CASP1CASP7KMT2A
SCHEMBL2425515 0.70 MAPT (0.43) MAPKAPK2CDK1MEN1KMT2APDE4B
SCHEMBL5230177 0.64 PARP1 (0.46) ALDH1A1PIM1CSNK2A1DYRK1ACLK4
SCHEMBL794250 0.63 PARP11 (0.44) PARP10PARP11PIM1CSNK2A1DYRK1A
SCHEMBL26512104 0.63 MAPKAPK2 (0.35) MAPKAPK2MKNK1MKNK2
SCHEMBL5320061 0.62 CYP1A2 (0.31)
SCHEMBL5393255 0.62 POLB (0.46) ALDH1A1PIM1CSNK2A1DYRK1ACLK4
SCHEMBL3794487 0.62 CYP1A2 (0.46) ALDH1A1MEN1KMT2ANPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1540329-A4 DRUG DISCOVERY METHOD KEDDEM BIO SCIENCE LTD (IL) 2009-06-10 EP disclosed
EP-1540329-A1 DRUG DISCOVERY METHOD KEDDEM BIO-SCIENCE LTD. (IL) 2005-06-15 EP disclosed
WO-2004010136-A1 DRUG DISCOVERY METHOD KEDDEM BIO-SCIENCE LTD. (IL) 2004-01-29 WO disclosed