Pyrene

Pyrene

SCHEMBL433757

c1cc2ccc3cccc4ccc(c1)c2c34.c1ccc2c(c1)ccc1cccnc12

nearest known ligand 0.60

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 3/20 0.60
MAPT P10636 5/20 0.58
SMN1; SMN2 Q16637 5/20 0.58
KDM4E B2RXH2 5/20 0.58
CYP3A4 P08684 4/20 0.58
CCR1 P32246 4/20 0.58
CCR8 P51685 4/20 0.58
TDP1 Q9NUW8 3/20 0.58
TSHR P16473 3/20 0.58
MMP2 P08253 2/20 0.58
TP53 P04637 2/20 0.58
CCR5 P51681 2/20 0.58
GMNN O75496 1/20 0.58
HSP90AA1 P07900 1/20 0.58
CYP2D6 P10635 1/20 0.58
MMP9 P14780 1/20 0.58
ALOX15 P16050 1/20 0.58
NFKB1 P19838 1/20 0.58
MMP8 P22894 1/20 0.58
THPO P40225 1/20 0.58

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
1-Naphthoquinoline SCHEMBL29533982 0.92 LMNA (0.69) LMNAMAPTSMN1; SMN2KDM4ECYP3A4
1-Naphthoquinoline SCHEMBL15106 0.92 LMNA (0.69) LMNAMAPTSMN1; SMN2KDM4ECYP3A4
1-Naphthoquinoline SCHEMBL3045500 0.90 LMNA (0.67) LMNAMAPTSMN1; SMN2KDM4ECYP3A4
1-Naphthoquinoline SCHEMBL31141994 0.90 LMNA (0.67) LMNAMAPTSMN1; SMN2KDM4ECYP3A4
1-Naphthoquinoline SCHEMBL31286254 0.90 LMNA (0.67) LMNAMAPTSMN1; SMN2KDM4ECYP3A4
1-Naphthoquinoline SCHEMBL6826374 0.90 LMNA (0.67) LMNAMAPTSMN1; SMN2KDM4ECYP3A4
1-Naphthoquinoline SCHEMBL5572864 0.90 LMNA (0.67) LMNAMAPTSMN1; SMN2KDM4ECYP3A4
1-Naphthoquinoline SCHEMBL6340901 0.90 LMNA (0.67) LMNAMAPTSMN1; SMN2KDM4ECYP3A4
SCHEMBL3193877 0.90 LMNA (0.67) LMNAMAPTSMN1; SMN2KDM4ECYP3A4
1-Naphthoquinoline SCHEMBL262791 0.90 LMNA (0.67) LMNAMAPTSMN1; SMN2KDM4ECYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 17 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20180005758-A1 USE OF ORGANIC AND ORGANOMETALLIC HIGH DIELECTRIC CONSTANT MATERIAL FOR IMPROVED ENERGY STORAGE DEVICES AND ASSOCIATED METHODS CLEANVOLT ENERGY, INC. 2018-01-04 US claimed
CN-103250216-B The application in the energy storing device improved of organic and organic metal high dielectric constant material and correlation technique CLEANVOLT ENERGY, INC. (US) 2016-02-24 CN claimed
US-20150162131-A1 USE OF ORGANIC AND ORGANOMETALLIC HIGH DIELECTRIC CONSTANT MATERIAL FOR IMPROVED ENERGY STORAGE DEVICES AND ASSOCIATED METHODS CLEANVOLT ENERGY, INC. 2015-06-11 US claimed
CN-103250216-A Use of organic and organometallic high dielectric constant material for improved energy storage devices and associated methods CLEANVOLT ENERGY INC 2013-08-14 CN claimed
US-20130194723-A1 USE OF ORGANIC AND ORGANOMETALLIC HIGH DIELECTRIC CONSTANT MATERIAL FOR IMPROVED ENERGY STORAGE DEVICES AND ASSOCIATED METHODS CLEANVOLT ENERGY, INC. (US) 2013-08-01 US claimed
EP-2596508-A2 USE OF ORGANIC AND ORGANOMETALLIC HIGH DIELECTRIC CONSTANT MATERIAL FOR IMPROVED ENERGY STORAGE DEVICES AND ASSOCIATED METHODS Cleanvolt Energy, Inc. (US) 2013-05-29 EP claimed
WO-2012012672-A2 USE OF ORGANIC AND ORGANOMETALLIC HIGH DIELECTRIC CONSTANT MATERIAL FOR IMPROVED ENERGY STORAGE DEVICES AND ASSOCIATED METHODS CLEANVOLT ENERGY, INC. (US) 2012-01-26 WO claimed
EP-2596508-B1 USE OF ORGANIC AND ORGANOMETALLIC HIGH DIELECTRIC CONSTANT MATERIAL FOR IMPROVED ENERGY STORAGE DEVICES AND ASSOCIATED METHODS CLEANVOLT ENERGY INC (US) 2024-05-22 EP disclosed
US-20180005758-A1 USE OF ORGANIC AND ORGANOMETALLIC HIGH DIELECTRIC CONSTANT MATERIAL FOR IMPROVED ENERGY STORAGE DEVICES AND ASSOCIATED METHODS CLEANVOLT ENERGY, INC. 2018-01-04 US disclosed
US-9767960-B2 Use of organic and organometallic high dielectric constant material for improved energy storage devices and associated methods CLEANVOLT ENERGY, INC. (US) 2017-09-19 US disclosed
CN-103250216-B The application in the energy storing device improved of organic and organic metal high dielectric constant material and correlation technique CLEANVOLT ENERGY, INC. (US) 2016-02-24 CN disclosed
US-20150162131-A1 USE OF ORGANIC AND ORGANOMETALLIC HIGH DIELECTRIC CONSTANT MATERIAL FOR IMPROVED ENERGY STORAGE DEVICES AND ASSOCIATED METHODS CLEANVOLT ENERGY, INC. 2015-06-11 US disclosed
US-8929054-B2 Use of organic and organometallic high dielectric constant material for improved energy storage devices and associated methods CLEANVOLT ENERGY, INC. (US) 2015-01-06 US disclosed
CN-103250216-A Use of organic and organometallic high dielectric constant material for improved energy storage devices and associated methods CLEANVOLT ENERGY INC 2013-08-14 CN disclosed
US-20130194723-A1 USE OF ORGANIC AND ORGANOMETALLIC HIGH DIELECTRIC CONSTANT MATERIAL FOR IMPROVED ENERGY STORAGE DEVICES AND ASSOCIATED METHODS CLEANVOLT ENERGY, INC. (US) 2013-08-01 US disclosed
EP-2596508-A2 USE OF ORGANIC AND ORGANOMETALLIC HIGH DIELECTRIC CONSTANT MATERIAL FOR IMPROVED ENERGY STORAGE DEVICES AND ASSOCIATED METHODS Cleanvolt Energy, Inc. (US) 2013-05-29 EP disclosed
WO-2012012672-A2 USE OF ORGANIC AND ORGANOMETALLIC HIGH DIELECTRIC CONSTANT MATERIAL FOR IMPROVED ENERGY STORAGE DEVICES AND ASSOCIATED METHODS CLEANVOLT ENERGY, INC. (US) 2012-01-26 WO disclosed