SCHEMBL4337706

SCHEMBL4337706

CC1(C)OCC(c2cc(F)cc(F)c2)N(C(=O)O)C1=O

nearest known ligand 0.36

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
RIPK1 Q13546 5/20 0.36
HCAR3 P49019 1/20 0.33
HCAR2 Q8TDS4 1/20 0.33
MDM2 Q00987 2/20 0.31
TP53 P04637 1/20 0.31
HTR7 P34969 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1274517 1.00 RIPK1 (0.36) RIPK1HCAR3HCAR2MDM2TP53
SCHEMBL1274826 0.82 RIPK1 (0.37) RIPK1HCAR3HCAR2MDM2TP53
SCHEMBL12311280 0.80 RIPK1 (0.33) RIPK1
SCHEMBL12263102 0.78 MDM2 (0.36) RIPK1MDM2TP53
SCHEMBL6961509 0.76 RIPK1 (0.37) RIPK1TP53HTR7
SCHEMBL1068636 0.71 RIPK1 (0.34) RIPK1MDM2TP53
SCHEMBL978138 0.71 RIPK1 (0.34) RIPK1MDM2TP53
SCHEMBL1272344 0.68 RIPK1 (0.38) RIPK1HTR7
SCHEMBL1274500 0.67 PGR (0.35)
SCHEMBL1273295 0.67 RIPK1 (0.41) RIPK1TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2024358-A1 SUBSTITUTED SPIROCYCLIC CGRP RECEPTOR ANTAGONISTS Merck & Co., Inc. (US) 2009-02-18 EP disclosed
WO-2007133491-A1 SUBSTITUTED SPIROCYCLIC CGRP RECEPTOR ANTAGONISTS MERCK & CO., INC. (US) 2007-11-22 WO disclosed