SCHEMBL4337980

SCHEMBL4337980

CC(=O)Oc1ccc2nc(Cl)ncc2c1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.55
GLA P06280 2/20 0.55
F2 P00734 1/20 0.55
HPGD P15428 1/20 0.55
PDE3B Q13370 1/20 0.49
PDE3A Q14432 1/20 0.49
KDM4E B2RXH2 4/20 0.44
SMN1; SMN2 Q16637 3/20 0.44
CA2 P00918 3/20 0.43
CA12 O43570 2/20 0.42
CA9 Q16790 2/20 0.42
FLT3 P36888 1/20 0.42
KMT2A Q03164 2/20 0.41
TUBB4A P04350 1/20 0.41
TUBB P07437 1/20 0.41
TUBA3C P0DPH7 1/20 0.41
TUBA1B P68363 1/20 0.41
TUBA4A P68366 1/20 0.41
TUBB4B P68371 1/20 0.41
TUBB3 Q13509 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27766565 0.88 ALDH1A1 (0.48) ALDH1A1GLAF2HPGDPDE3B
SCHEMBL27801346 0.83 GLA (0.56) ALDH1A1GLAF2HPGDPDE3B
SCHEMBL3719415 0.81 ALDH1A1 (0.46) ALDH1A1HPGDPDE3BPDE3AKDM4E
SCHEMBL1571317 0.79 ALDH1A1 (0.59) ALDH1A1GLAF2HPGDPDE3B
SCHEMBL28814899 0.79 ALDH1A1 (0.67) ALDH1A1GLAF2HPGDPDE3B
SCHEMBL27929529 0.78 PDE3B (0.51) ALDH1A1GLAF2HPGDPDE3B
Hydrochloric Acid SCHEMBL28007029 0.78 ALDH1A1 (0.57) ALDH1A1GLAF2HPGDPDE3B
SCHEMBL535665 0.77 EGFR (0.64) ALDH1A1GLAF2HPGDPDE3B
SCHEMBL4857055 0.76 KMT2A (0.53) ALDH1A1HPGDPDE3BPDE3AKDM4E
Hydrochloric Acid SCHEMBL30406782 0.76 EGFR (0.62) ALDH1A1GLAF2HPGDPDE3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101652352-A Quinazolines for PDK1 inhibition NOVARTIS VACCINES & DIAGNOSTIC 2010-02-17 CN disclosed
EP-2061772-A2 MULTI-FUNCTIONAL SMALL MOLECULES AS ANTI-PROLIFERATIVE AGENTS Curis, Inc. (US) 2009-05-27 EP disclosed
WO-2008033747-A9 MULTI-FUNCTIONAL SMALL MOLECULES AS ANTI-PROLIFERATIVE AGENTS CURIS INC (MA) 2008-07-24 WO disclosed
WO-2008033747-A2 MULTI-FUNCTIONAL SMALL MOLECULES AS ANTI-PROLIFERATIVE AGENTS CURIS, INC. (US) 2008-03-20 WO disclosed
US-5932574-A ANTICANCER AGENT ZENECA LIMITED (GB) 1999-08-03 US disclosed