SCHEMBL434008

SCHEMBL434008

Cc1noc2ccc(C3(C(=O)NC(CN4CCCC4)c4ccccc4)CC3)cc12

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNK3 O14649 5/20 0.40
ROCK2 O75116 1/20 0.38
ROCK1 Q13464 1/20 0.38
GPR88 Q9GZN0 1/20 0.37
RPS6KB1 P23443 2/20 0.37
AURKA O14965 1/20 0.37
AURKB Q96GD4 1/20 0.37
TAS2R8 Q9NYW2 1/20 0.36
MAPK1 P28482 2/20 0.36
NPC1 O15118 1/20 0.35
ALDH1A1 P00352 1/20 0.35
SMYD3 Q9H7B4 1/20 0.35
ABCC3 O15438 1/20 0.35
ABCC4 O15439 1/20 0.35
ABCB11 O95342 1/20 0.35
CYP2C8 P10632 1/20 0.35
CYP2C9 P11712 1/20 0.35
ABCB4 P21439 1/20 0.35
LPAR1 Q92633 1/20 0.35
ABCC2 Q92887 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15385517 1.00 KCNK3 (0.40) KCNK3ROCK2ROCK1GPR88RPS6KB1
SCHEMBL433254 0.83 MAPK1 (0.42) ROCK2ROCK1GPR88AURKAAURKB
SCHEMBL433255 0.83 MAPK1 (0.42) ROCK2ROCK1GPR88AURKAAURKB
SCHEMBL10083742 0.81 ROCK2 (0.41) KCNK3ROCK2ROCK1GPR88RPS6KB1
SCHEMBL434527 0.81 ROCK2 (0.41) KCNK3ROCK2ROCK1GPR88RPS6KB1
SCHEMBL10084059 0.81 HDAC4 (0.49) KCNK3ROCK2ROCK1GPR88RPS6KB1
SCHEMBL435831 0.80 HSD11B1 (0.50) GPR88MAPK1NPC1ALDH1A1
SCHEMBL15385492 0.80 HSD11B1 (0.50) GPR88MAPK1NPC1ALDH1A1
Hydrochloric Acid SCHEMBL459715 0.80 HDAC4 (0.48) ROCK2ROCK1GPR88NPC1ALDH1A1
Hydrochloric Acid SCHEMBL15380914 0.80 HDAC4 (0.48) ROCK2ROCK1GPR88NPC1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012012410-A2 KAPPA OPIOID RECEPTOR AGONISTS DR. REDDY'S LABORATORIES LTD. (IN) 2012-01-26 WO disclosed