SCHEMBL4342196

SCHEMBL4342196

CC(O)c1cc(NC(=O)N(S)Cc2ccccc2)cc(Cl)c1O

nearest known ligand 0.42

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
EGFR P00533 4/20 0.41
ERBB2 P04626 4/20 0.41
ALDH1A1 P00352 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
UBE2M P61081 3/20 0.39
DCUN1D1 Q96GG9 3/20 0.39
HTT P42858 2/20 0.38
GAA P10253 2/20 0.38
LMNA P02545 1/20 0.38
DHODH Q02127 1/20 0.38
MTOR P42345 1/20 0.38
MEN1 O00255 1/20 0.37
KMT2A Q03164 1/20 0.37
TDP1 Q9NUW8 1/20 0.37
RORC P51449 1/20 0.37
CYP1A2 P05177 1/20 0.37
CYP2C9 P11712 1/20 0.37
CYP2C19 P33261 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4355801 0.87 EGFR (0.48) EGFRERBB2ALDH1A1NPSR1UBE2M
SCHEMBL4351073 0.82 HTT (0.40) EGFRERBB2NPSR1UBE2MDCUN1D1
SCHEMBL4342217 0.78 EGFR (0.38) EGFRERBB2UBE2MDCUN1D1GAA
SCHEMBL4349798 0.77 ALDH1A1 (0.46) EGFRERBB2ALDH1A1NPSR1UBE2M
SCHEMBL4341765 0.77 KMT2A (0.54) NPSR1HTTGAALMNADHODH
SCHEMBL4349474 0.76 EPHX1 (0.58) ALDH1A1HTTLMNAMEN1KMT2A
SCHEMBL4349894 0.76 GAA (0.40) ALDH1A1HTTGAALMNADHODH
SCHEMBL4354101 0.76 SMN1; SMN2 (0.39) EGFRERBB2ALDH1A1HTTGAA
SCHEMBL4345339 0.76 ALDH1A1 (0.49) EGFRERBB2ALDH1A1NPSR1UBE2M
SCHEMBL4345437 0.74 EGFR (0.48) EGFRERBB2ALDH1A1NPSR1MTOR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2100876-A2 New compounds for the inhibition of rotamases and use thereof Jerini AG (DE) 2009-09-16 EP claimed
EP-2100876-A2 New compounds for the inhibition of rotamases and use thereof Jerini AG (DE) 2009-09-16 EP disclosed