SCHEMBL4354101

SCHEMBL4354101

CC(O)c1cc(N(S)C(=O)Nc2ccccc2)cc(Cl)c1O

nearest known ligand 0.39

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 3/20 0.39
NPC1 O15118 2/20 0.39
MAPT P10636 2/20 0.39
HSD17B10 Q99714 2/20 0.39
ALDH1A1 P00352 1/20 0.39
ALOX15 P16050 1/20 0.39
RAB9A P51151 1/20 0.39
MTOR P42345 1/20 0.39
BCL2 P10415 1/20 0.39
EGFR P00533 4/20 0.39
ERBB2 P04626 3/20 0.39
STK39 Q9UEW8 1/20 0.38
MEN1 O00255 2/20 0.37
KMT2A Q03164 2/20 0.37
NPY5R Q15761 2/20 0.37
LMNA P02545 2/20 0.36
HTT P42858 2/20 0.36
GAA P10253 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4355433 0.91 TSHR (0.43) SMN1; SMN2NPC1MAPTHSD17B10ALDH1A1
SCHEMBL4354080 0.87 ALDH1A1 (0.36) SMN1; SMN2MAPTALDH1A1RAB9ASTK39
SCHEMBL4351896 0.86 MAPT (0.48) SMN1; SMN2NPC1MAPTHSD17B10ALDH1A1
SCHEMBL4348453 0.85 PDE2A (0.42) SMN1; SMN2MTORLMNAHTT
SCHEMBL4349857 0.82 POLB (0.41) SMN1; SMN2NPC1ALDH1A1RAB9AMEN1
SCHEMBL4351937 0.81 MAPK1 (0.33) MAPTALDH1A1MEN1KMT2AGAA
SCHEMBL4350109 0.81 CA1 (0.41) SMN1; SMN2NPC1ALDH1A1RAB9AMEN1
SCHEMBL4344614 0.81 MAPT (0.40) SMN1; SMN2NPC1MAPTHSD17B10ALDH1A1
SCHEMBL4345462 0.78 NPC1 (0.39) NPC1ALDH1A1RAB9AKMT2ALMNA
SCHEMBL4341765 0.77 KMT2A (0.54) SMN1; SMN2NPC1MAPTHSD17B10RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2100876-A2 New compounds for the inhibition of rotamases and use thereof Jerini AG (DE) 2009-09-16 EP claimed
EP-2100876-A2 New compounds for the inhibition of rotamases and use thereof Jerini AG (DE) 2009-09-16 EP disclosed