SCHEMBL4342197

SCHEMBL4342197

Oc1ccc(NC(=S)Nc2ccc(C(F)(F)F)cc2)cc1F

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK1 P06493 1/20 0.51
MEN1 O00255 6/20 0.51
KMT2A Q03164 6/20 0.51
CA12 O43570 1/20 0.50
CA1 P00915 1/20 0.50
CA2 P00918 1/20 0.50
CA9 Q16790 1/20 0.50
MAPT P10636 7/20 0.48
ALDH1A1 P00352 4/20 0.48
SMN1; SMN2 Q16637 3/20 0.48
HTT P42858 3/20 0.48
KDM4E B2RXH2 3/20 0.48
GAA P10253 3/20 0.48
LMNA P02545 2/20 0.48
KIF11 P52732 1/20 0.47
HSPA9 P38646 1/20 0.47
NPSR1 Q6W5P4 4/20 0.47
L3MBTL1 Q9Y468 1/20 0.47
TDP1 Q9NUW8 2/20 0.46
EPHX2 P34913 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4358929 0.86 CDK1 (0.53) CDK1MEN1KMT2ACA12CA1
SCHEMBL4354013 0.85 MEN1 (0.64) CDK1MEN1KMT2AMAPTALDH1A1
SCHEMBL4341318 0.83 MAPT (0.59) CDK1MEN1KMT2ACA12CA1
SCHEMBL9453957 0.83 CDK1 (0.68) CDK1MEN1KMT2ACA12CA1
SCHEMBL4345620 0.82 KMT2A (0.59) MEN1KMT2AMAPTALDH1A1SMN1; SMN2
SCHEMBL4348076 0.81 MEN1 (0.62) MEN1KMT2AMAPTALDH1A1SMN1; SMN2
SCHEMBL18031170 0.80 GAA (0.69) CDK1MEN1KMT2ACA12CA1
SCHEMBL4350936 0.79 KMT2A (0.62) MEN1KMT2AMAPTALDH1A1SMN1; SMN2
SCHEMBL4345484 0.77 HRAS (0.54) CDK1MEN1KMT2ACA12CA1
SCHEMBL4353931 0.77 TMPRSS4 (0.58) CDK1MEN1KMT2AMAPTALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-100546977-C Suppress the new compound and the application thereof of rotamase JERINI AG (DE) 2009-10-07 CN claimed
EP-2100876-A2 New compounds for the inhibition of rotamases and use thereof Jerini AG (DE) 2009-09-16 EP claimed
CN-1701061-A Novel compounds for inhibiting rotamase enzymes and uses thereof JERINI AG (DE) 2005-11-23 CN claimed
EP-2100876-A2 New compounds for the inhibition of rotamases and use thereof Jerini AG (DE) 2009-09-16 EP disclosed