SCHEMBL4345484

SCHEMBL4345484

O=[N+]([O-])c1cc(NC(=S)Nc2ccc(C(F)(F)F)cc2)ccc1O

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HRAS P01112 2/20 0.54
MAPT P10636 6/20 0.50
GAA P10253 4/20 0.50
MEN1 O00255 3/20 0.50
KMT2A Q03164 3/20 0.50
HTT P42858 2/20 0.50
SMN1; SMN2 Q16637 2/20 0.50
LMNA P02545 1/20 0.50
ALOX12 P18054 1/20 0.50
CA12 O43570 2/20 0.49
CA1 P00915 2/20 0.49
CA2 P00918 2/20 0.49
CA9 Q16790 2/20 0.49
ALDH1A1 P00352 5/20 0.48
HPGD P15428 2/20 0.48
PPIA P62937 1/20 0.48
NPSR1 Q6W5P4 3/20 0.47
NPY1R P25929 1/20 0.47
NPY2R P49146 1/20 0.47
HSPA9 P38646 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4347085 0.88 CA12 (0.61) MAPTGAAMEN1KMT2AHTT
SCHEMBL4341575 0.87 MEN1 (0.59) HRASMAPTGAAMEN1KMT2A
SCHEMBL4353650 0.83 MAPT (0.63) MAPTGAAMEN1KMT2AHTT
SCHEMBL4346971 0.82 PPIA (0.58) MAPTGAAMEN1KMT2AHTT
SCHEMBL4357616 0.82 ALDH1A1 (0.63) MAPTGAAMEN1KMT2AHTT
SCHEMBL4345759 0.80 ALDH1A1 (0.51) MAPTGAAMEN1KMT2AHTT
SCHEMBL4344002 0.78 PPIA (0.56) MAPTGAAMEN1KMT2AHTT
SCHEMBL4346879 0.78 MTOR (0.62) GAAMEN1KMT2ACA12CA1
SCHEMBL1026402 0.78 ALDH1A1 (0.56) MAPTMEN1KMT2ASMN1; SMN2LMNA
SCHEMBL4342197 0.77 CDK1 (0.51) MAPTGAAMEN1KMT2AHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-100546977-C Suppress the new compound and the application thereof of rotamase JERINI AG (DE) 2009-10-07 CN claimed
EP-2100876-A2 New compounds for the inhibition of rotamases and use thereof Jerini AG (DE) 2009-09-16 EP claimed
CN-1701061-A Novel compounds for inhibiting rotamase enzymes and uses thereof JERINI AG (DE) 2005-11-23 CN claimed
EP-2100876-A2 New compounds for the inhibition of rotamases and use thereof Jerini AG (DE) 2009-09-16 EP disclosed