SCHEMBL4354013

SCHEMBL4354013

Oc1ccc(NC(=S)NCc2ccc(C(F)(F)F)cc2)cc1F

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 9/20 0.64
KMT2A Q03164 9/20 0.64
MAPT P10636 8/20 0.64
ALDH1A1 P00352 6/20 0.64
GAA P10253 3/20 0.64
SMN1; SMN2 Q16637 2/20 0.64
LMNA P02545 6/20 0.60
HPGD P15428 3/20 0.60
NPSR1 Q6W5P4 2/20 0.60
L3MBTL1 Q9Y468 1/20 0.60
MAPK1 P28482 1/20 0.60
HTT P42858 3/20 0.56
MYC P01106 1/20 0.55
MAX P61244 1/20 0.55
CDK1 P06493 1/20 0.50
ALOX12 P18054 1/20 0.50
BLM P54132 1/20 0.50
MTOR P42345 1/20 0.49
DUSP3 P51452 1/20 0.48
MAOA P21397 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4341860 0.87 MEN1 (0.63) MEN1KMT2AMAPTALDH1A1GAA
SCHEMBL4357659 0.86 MAPT (0.62) MEN1KMT2AMAPTALDH1A1GAA
SCHEMBL4342197 0.85 CDK1 (0.51) MEN1KMT2AMAPTALDH1A1GAA
SCHEMBL4347646 0.85 MTOR (0.70) MEN1KMT2ASMN1; SMN2LMNAMTOR
SCHEMBL4343714 0.84 RAB9A (0.63) MEN1KMT2AMAPTALDH1A1GAA
SCHEMBL4341575 0.81 MEN1 (0.59) MEN1KMT2AMAPTALDH1A1GAA
SCHEMBL28034498 0.78 MAPT (0.89) MEN1KMT2AMAPTALDH1A1GAA
SCHEMBL18695140 0.78 MAPT (1.00) MEN1KMT2AMAPTALDH1A1GAA
SCHEMBL4351636 0.78 MEN1 (0.61) MEN1KMT2AMAPTALDH1A1GAA
SCHEMBL4357497 0.78 MEN1 (0.61) MEN1KMT2AMAPTALDH1A1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-100546977-C Suppress the new compound and the application thereof of rotamase JERINI AG (DE) 2009-10-07 CN claimed
EP-2100876-A2 New compounds for the inhibition of rotamases and use thereof Jerini AG (DE) 2009-09-16 EP claimed
CN-1701061-A Novel compounds for inhibiting rotamase enzymes and uses thereof JERINI AG (DE) 2005-11-23 CN claimed
EP-2100876-A2 New compounds for the inhibition of rotamases and use thereof Jerini AG (DE) 2009-09-16 EP disclosed