SCHEMBL4344004

SCHEMBL4344004

O=C(Nc1ccc(O)c([N+](=O)[O-])c1)N(S)c1cc(Cl)cc(Cl)c1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
P2RX1 P51575 2/20 0.48
MEN1 O00255 3/20 0.41
KMT2A Q03164 3/20 0.41
HTT P42858 3/20 0.41
LMNA P02545 2/20 0.41
MAPT P10636 2/20 0.41
GAA P10253 1/20 0.41
EGFR P00533 1/20 0.41
AURKB Q96GD4 1/20 0.41
ALDH5A1 P51649 1/20 0.40
ABAT P80404 1/20 0.40
SMN1; SMN2 Q16637 2/20 0.39
MAPK1 P28482 2/20 0.39
ALDH1A1 P00352 1/20 0.39
TP53 P04637 1/20 0.39
HPGD P15428 1/20 0.39
TSHR P16473 1/20 0.39
GPR35 Q9HC97 1/20 0.39
DHODH Q02127 1/20 0.39
TTR P02766 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4346974 0.90 P2RX1 (0.51) P2RX1MEN1KMT2AHTTLMNA
SCHEMBL4342020 0.79 MAPT (0.57) P2RX1MEN1KMT2AHTTLMNA
SCHEMBL4353654 0.78 MAPT (0.49) MEN1KMT2AHTTLMNAMAPT
SCHEMBL10882608 0.76 APEX1 (0.50) P2RX1MEN1KMT2AHTTLMNA
SCHEMBL4345763 0.76 MAPK1 (0.43) P2RX1MEN1KMT2AHTTLMNA
SCHEMBL4344002 0.76 PPIA (0.56) P2RX1MEN1KMT2AHTTLMNA
SCHEMBL4345489 0.75 CA12 (0.47) P2RX1MEN1KMT2ALMNAMAPT
SCHEMBL4356349 0.75 MEN1 (0.62) P2RX1MEN1KMT2AHTTLMNA
SCHEMBL6975312 0.72 MAPT (0.54) P2RX1MEN1KMT2AHTTLMNA
SCHEMBL6975308 0.72 MAPT (0.54) P2RX1MEN1KMT2AHTTLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2100876-A2 New compounds for the inhibition of rotamases and use thereof Jerini AG (DE) 2009-09-16 EP claimed
EP-2100876-A2 New compounds for the inhibition of rotamases and use thereof Jerini AG (DE) 2009-09-16 EP disclosed