SCHEMBL4344002

SCHEMBL4344002

O=[N+]([O-])c1cc(NC(=S)Nc2cc(Cl)cc(Cl)c2)ccc1O

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PPIA P62937 1/20 0.56
MEN1 O00255 3/20 0.52
KMT2A Q03164 3/20 0.52
P2RX1 P51575 1/20 0.50
MAOB P27338 1/20 0.50
ALDH1A1 P00352 6/20 0.47
MAPT P10636 4/20 0.47
HPGD P15428 3/20 0.47
GAA P10253 2/20 0.47
SMN1; SMN2 Q16637 2/20 0.47
HTT P42858 1/20 0.47
DHODH Q02127 1/20 0.45
EGFR P00533 1/20 0.45
LMNA P02545 1/20 0.44
POLB P06746 1/20 0.44
NPSR1 Q6W5P4 1/20 0.44
ALDH5A1 P51649 1/20 0.44
ABAT P80404 1/20 0.44
IDO1 P14902 1/20 0.44
TP53 P04637 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4346971 0.90 PPIA (0.58) PPIAMEN1KMT2AP2RX1ALDH1A1
SCHEMBL4342020 0.87 MAPT (0.57) MEN1KMT2AP2RX1MAPTGAA
SCHEMBL4353650 0.83 MAPT (0.63) PPIAMEN1KMT2AMAOBALDH1A1
SCHEMBL30542217 0.80 ALDH1A1 (0.62) MEN1KMT2AMAOBALDH1A1MAPT
SCHEMBL4345759 0.79 ALDH1A1 (0.51) PPIAMEN1KMT2AALDH1A1MAPT
SCHEMBL4345484 0.78 HRAS (0.54) PPIAMEN1KMT2AALDH1A1MAPT
SCHEMBL28529066 0.78 MAPK1 (0.53) PPIAMEN1KMT2AP2RX1ALDH1A1
SCHEMBL4357526 0.78 ALDH1A1 (0.50) PPIAMEN1KMT2AALDH1A1MAPT
SCHEMBL4341617 0.77 MAOB (0.60) MEN1KMT2AMAOBALDH1A1MAPT
SCHEMBL4356349 0.77 MEN1 (0.62) MEN1KMT2AP2RX1MAPTGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2100876-A2 New compounds for the inhibition of rotamases and use thereof Jerini AG (DE) 2009-09-16 EP claimed
CN-1701061-A Novel compounds for inhibiting rotamase enzymes and uses thereof JERINI AG (DE) 2005-11-23 CN claimed
EP-2100876-A2 New compounds for the inhibition of rotamases and use thereof Jerini AG (DE) 2009-09-16 EP disclosed