SCHEMBL4344179

SCHEMBL4344179

Clc1cccc(C(C(c2cccnc2)c2cccnc2)N2CCOCC2)c1Cl

nearest known ligand 0.53

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
P2RX7 Q99572 5/20 0.53
KCNA5 P22460 4/20 0.48
POLB P06746 4/20 0.43
ALDH1A1 P00352 4/20 0.43
KDM4E B2RXH2 3/20 0.43
HSD17B10 Q99714 1/20 0.41
GAA P10253 1/20 0.41
LMNA P02545 1/20 0.41
TP53 P04637 1/20 0.41
MAPT P10636 1/20 0.41
DPP4 P27487 1/20 0.40
KCNH2 Q12809 1/20 0.40
CYP3A4 P08684 1/20 0.39
CYP2C9 P11712 1/20 0.39
CYP2C19 P33261 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1240803 0.82 KCNA5 (0.52) P2RX7KCNA5POLBALDH1A1KDM4E
SCHEMBL1243292 0.81 POLB (0.54) P2RX7KCNA5POLBALDH1A1KDM4E
SCHEMBL1242829 0.80 P2RX7 (0.46) P2RX7KCNA5POLBALDH1A1KDM4E
SCHEMBL1243271 0.79 ALDH1A1 (0.47) P2RX7KCNA5POLBALDH1A1KDM4E
SCHEMBL12194951 0.78 KCNA5 (0.67) P2RX7KCNA5POLB
SCHEMBL1242284 0.76 KCNA5 (0.47) P2RX7KCNA5POLBALDH1A1KDM4E
SCHEMBL1242866 0.75 MAPT (0.51) KCNA5POLBALDH1A1KDM4EHSD17B10
SCHEMBL1242030 0.75 KCNA5 (0.49) KCNA5POLBALDH1A1KDM4EHSD17B10
SCHEMBL1242226 0.74 KCNA5 (0.45) KCNA5POLBALDH1A1KDM4EHSD17B10
SCHEMBL2473671 0.74 KCNA5 (0.46) P2RX7KCNA5POLBALDH1A1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1781635-A4 POTASSIUM CHANNEL INHIBITORS MERCK & CO INC (US) 2009-02-25 EP disclosed
EP-1781635-A2 POTASSIUM CHANNEL INHIBITORS Merck & Co., Inc. (US) 2007-05-09 EP disclosed
WO-2006015159-A2 POTASSIUM CHANNEL INHIBITORS MERCK & CO., INC. (US) 2006-02-09 WO disclosed