SCHEMBL4344872

SCHEMBL4344872

CC(C)(C)[C@H](NC(=O)c1cc2cc(F)ccc2[nH]1)C(=O)N1C[C@@H]2C[C@H]1CN2C(=O)[C@H]1COCCN1S(=O)(=O)c1cc(C(F)(F)F)ccc1Cl

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMYD3 Q9H7B4 2/20 0.37
HCRTR1 O43613 2/20 0.36
HCRTR2 O43614 2/20 0.36
CYP51A1 Q16850 3/20 0.34
STAT6 P42226 2/20 0.34
PYGL P06737 1/20 0.34
PYGM P11217 1/20 0.34
HSD11B1 P28845 2/20 0.33
MCHR1 Q99705 1/20 0.33
KDM4E B2RXH2 1/20 0.32
ALDH1A1 P00352 1/20 0.32
LMNA P02545 1/20 0.32
GAA P10253 1/20 0.32
MAPT P10636 1/20 0.32
LGALS8 O00214 1/20 0.32
LGALS3 P17931 1/20 0.32
MLLT1 Q03111 1/20 0.32
DRD2 P14416 1/20 0.31
DRD3 P35462 1/20 0.31
HRH4 Q9H3N8 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19856901 0.87 STAT6 (0.38) SMYD3CYP51A1STAT6PYGLPYGM
SCHEMBL19856903 0.87 STAT6 (0.38) SMYD3CYP51A1STAT6PYGLPYGM
SCHEMBL4343724 0.86 CYP51A1 (0.36) SMYD3CYP51A1STAT6PYGLPYGM
SCHEMBL19856965 0.85 TDP1 (0.36) SMYD3CYP51A1STAT6PYGLKDM4E
SCHEMBL4335350 0.85 TDP1 (0.36) SMYD3CYP51A1STAT6PYGLKDM4E
SCHEMBL19856915 0.85 TDP1 (0.36) SMYD3CYP51A1STAT6PYGLKDM4E
SCHEMBL4343721 0.85 TDP1 (0.36) SMYD3CYP51A1STAT6PYGLKDM4E
SCHEMBL19857011 0.84 SMYD3 (0.37) SMYD3HCRTR1HCRTR2CYP51A1STAT6
SCHEMBL4350449 0.81 HTRA1 (0.36) SMYD3CYP51A1STAT6PYGLKDM4E
SCHEMBL4341332 0.81 HTRA1 (0.36) SMYD3CYP51A1STAT6PYGLKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009146182-A1 TRPV4 ANTAGONISTS SMITHKLINE BEECHAM CORPORATION (US) 2009-12-03 WO claimed
WO-2009146182-A1 TRPV4 ANTAGONISTS SMITHKLINE BEECHAM CORPORATION (US) 2009-12-03 WO disclosed