SCHEMBL4345574

SCHEMBL4345574

O=[N+]([O-])c1cc(NCc2ccccc2Sc2ccc(Cl)cc2)cc(F)c1O

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.49
MAPT P10636 3/20 0.49
ALDH3A1 P30838 1/20 0.49
POLB P06746 2/20 0.47
GAA P10253 2/20 0.46
PKM P14618 1/20 0.46
SLC6A4 P31645 2/20 0.43
PDE7A Q13946 3/20 0.42
PDE7B Q9NP56 2/20 0.42
MEN1 O00255 2/20 0.41
KMT2A Q03164 2/20 0.41
MAPK1 P28482 1/20 0.41
BCL2L1 Q07817 2/20 0.40
PLA2G4A P47712 1/20 0.40
L3MBTL1 Q9Y468 2/20 0.39
IDO1 P14902 1/20 0.39
CYP1A2 P05177 1/20 0.39
CYP2C9 P11712 1/20 0.39
HPGD P15428 1/20 0.39
CYP2C19 P33261 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4345667 0.92 ALDH3A1 (0.50) ALDH1A1MAPTALDH3A1POLBGAA
SCHEMBL4349134 0.91 ALDH3A1 (0.47) ALDH1A1MAPTALDH3A1POLBGAA
SCHEMBL4345358 0.90 MAPT (0.47) ALDH1A1MAPTALDH3A1POLBGAA
SCHEMBL4346299 0.90 MAPT (0.47) ALDH1A1MAPTALDH3A1POLBGAA
SCHEMBL4342105 0.90 ALDH3A1 (0.47) ALDH1A1MAPTALDH3A1POLBGAA
SCHEMBL4342281 0.88 MAPT (0.46) ALDH1A1MAPTALDH3A1POLBGAA
SCHEMBL4346171 0.88 ALDH1A1 (0.51) ALDH1A1MAPTALDH3A1POLBGAA
SCHEMBL4354120 0.87 GAA (0.51) ALDH1A1MAPTALDH3A1POLBGAA
SCHEMBL4346420 0.87 PDE7A (0.48) ALDH1A1MAPTALDH3A1POLBGAA
SCHEMBL4347073 0.87 MEN1 (0.49) ALDH1A1MAPTPOLBGAAPKM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2100876-A2 New compounds for the inhibition of rotamases and use thereof Jerini AG (DE) 2009-09-16 EP claimed
CN-1701061-A Novel compounds for inhibiting rotamase enzymes and uses thereof JERINI AG (DE) 2005-11-23 CN claimed
WO-2004030664-A2 NEW COMPOUNDS FOR THE INHIBITION OF UNDESIRED CELL PROLIFERATION AND USE THEREOF JERINI AG (DE) 2004-04-15 WO claimed
EP-2100876-A2 New compounds for the inhibition of rotamases and use thereof Jerini AG (DE) 2009-09-16 EP disclosed