SCHEMBL4345899

SCHEMBL4345899

Oc1c(Cl)cc(NCc2ccccc2Sc2ccc(Cl)c(Cl)c2)cc1Cl

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 3/20 0.47
KMT2A Q03164 3/20 0.47
L3MBTL1 Q9Y468 2/20 0.47
MAPT P10636 2/20 0.47
ATM Q13315 1/20 0.47
HTR1A P08908 1/20 0.41
HTR3A P46098 1/20 0.41
CYP2C9 P11712 3/20 0.38
CYP2C19 P33261 3/20 0.38
CYP1A2 P05177 2/20 0.38
CYP3A4 P08684 2/20 0.38
PLA2G1B P04054 1/20 0.38
CYP2D6 P10635 1/20 0.38
ATG4B Q9Y4P1 1/20 0.38
MAOB P27338 2/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
ALDH1A1 P00352 1/20 0.37
HPGD P15428 1/20 0.37
GRM5 P41594 1/20 0.36
KDM4E B2RXH2 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6226736 0.90 MEN1 (0.41) MEN1KMT2AL3MBTL1MAPTATM
SCHEMBL4348016 0.89 MEN1 (0.41) MEN1KMT2AL3MBTL1MAPTATM
SCHEMBL4342244 0.89 MEN1 (0.50) MEN1KMT2AL3MBTL1MAPTATM
SCHEMBL4349840 0.88 SLC6A4 (0.48) MEN1KMT2AL3MBTL1MAPTATM
SCHEMBL4351063 0.88 SMN1; SMN2 (0.43) MEN1KMT2AL3MBTL1MAPTATM
SCHEMBL4355882 0.88 MEN1 (0.39) MEN1KMT2AL3MBTL1MAPTATM
SCHEMBL4348911 0.88 MEN1 (0.39) MEN1KMT2AL3MBTL1MAPTATM
SCHEMBL4345390 0.88 MAPT (0.51) MEN1KMT2AL3MBTL1MAPTATM
SCHEMBL4349243 0.86 MAPT (0.46) MEN1KMT2AL3MBTL1MAPTATM
SCHEMBL4354940 0.86 SLC6A4 (0.52) MEN1KMT2AL3MBTL1MAPTATM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2100876-A2 New compounds for the inhibition of rotamases and use thereof Jerini AG (DE) 2009-09-16 EP claimed
CN-1701061-A Novel compounds for inhibiting rotamase enzymes and uses thereof JERINI AG (DE) 2005-11-23 CN claimed
WO-2004030664-A2 NEW COMPOUNDS FOR THE INHIBITION OF UNDESIRED CELL PROLIFERATION AND USE THEREOF JERINI AG (DE) 2004-04-15 WO claimed
EP-2100876-A2 New compounds for the inhibition of rotamases and use thereof Jerini AG (DE) 2009-09-16 EP disclosed