SCHEMBL4354940

SCHEMBL4354940

Oc1c(Cl)cc(NCc2ccccc2Sc2cccc(Cl)c2)cc1Cl

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A4 P31645 2/20 0.52
SLC6A2 P23975 1/20 0.52
SLC6A3 Q01959 1/20 0.52
SMN1; SMN2 Q16637 1/20 0.42
CYP2C9 P11712 3/20 0.40
CYP2C19 P33261 3/20 0.40
MAPT P10636 3/20 0.40
CYP3A4 P08684 2/20 0.40
MEN1 O00255 2/20 0.40
KMT2A Q03164 2/20 0.40
KDM4E B2RXH2 1/20 0.40
ALOX15 P16050 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40
CYP1A2 P05177 2/20 0.40
PLA2G1B P04054 1/20 0.40
CYP2D6 P10635 1/20 0.40
ATG4B Q9Y4P1 1/20 0.40
L3MBTL1 Q9Y468 2/20 0.39
ALDH1A1 P00352 1/20 0.39
HPGD P15428 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6230536 0.90 SLC6A4 (0.46) SLC6A4SLC6A2SLC6A3SMN1; SMN2CYP2C9
SCHEMBL4351063 0.90 SMN1; SMN2 (0.43) SLC6A4SLC6A2SLC6A3SMN1; SMN2CYP2C9
SCHEMBL4351669 0.88 SLC6A4 (0.46) SLC6A4SLC6A2SLC6A3SMN1; SMN2CYP2C9
SCHEMBL4354464 0.88 SLC6A2 (0.46) SLC6A4SLC6A2SLC6A3SMN1; SMN2CYP2C9
SCHEMBL4351152 0.88 SLC6A4 (0.50) SLC6A4SLC6A2SLC6A3SMN1; SMN2CYP2C9
SCHEMBL4351653 0.88 SLC6A4 (0.53) SLC6A4SLC6A2SLC6A3SMN1; SMN2CYP2C9
SCHEMBL4345562 0.88 SLC6A2 (0.50) SLC6A4SLC6A2SLC6A3SMN1; SMN2CYP2C9
SCHEMBL4349840 0.87 SLC6A4 (0.48) SLC6A4SLC6A2SLC6A3SMN1; SMN2CYP2C9
SCHEMBL12846505 0.86 SLC6A4 (0.51) SLC6A4SLC6A2SLC6A3SMN1; SMN2CYP2C9
SCHEMBL4345899 0.86 MEN1 (0.47) SLC6A4SLC6A2SLC6A3SMN1; SMN2CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2100876-A2 New compounds for the inhibition of rotamases and use thereof Jerini AG (DE) 2009-09-16 EP claimed
CN-1701061-A Novel compounds for inhibiting rotamase enzymes and uses thereof JERINI AG (DE) 2005-11-23 CN claimed
WO-2004030664-A2 NEW COMPOUNDS FOR THE INHIBITION OF UNDESIRED CELL PROLIFERATION AND USE THEREOF JERINI AG (DE) 2004-04-15 WO claimed
EP-2100876-A2 New compounds for the inhibition of rotamases and use thereof Jerini AG (DE) 2009-09-16 EP disclosed