SCHEMBL4346161

SCHEMBL4346161

O=C(O)c1cc(NCc2ccccc2Sc2ccc(Cl)c(Cl)c2)ccc1O

nearest known ligand 0.60

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
NOX4 Q9NPH5 3/20 0.60
EGFR P00533 8/20 0.51
MAPT P10636 2/20 0.51
RGS12 O14924 1/20 0.51
ALDH1A1 P00352 1/20 0.51
LCK P06239 1/20 0.51
CAMKK2 Q96RR4 1/20 0.51
TDP1 Q9NUW8 1/20 0.51
KDM4C Q9H3R0 3/20 0.49
MEN1 O00255 1/20 0.43
KMT2A Q03164 1/20 0.43
ATM Q13315 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
PPARA Q07869 1/20 0.42
STING1 Q86WV6 1/20 0.42
PTPRG P23470 1/20 0.42
SYK P43405 2/20 0.42
SMN1; SMN2 Q16637 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4345406 0.89 NOX4 (0.62) NOX4EGFRMAPTRGS12ALDH1A1
SCHEMBL4358462 0.88 NOX4 (0.70) NOX4EGFRMAPTRGS12ALDH1A1
SCHEMBL4355493 0.87 NOX4 (0.60) NOX4EGFRMAPTRGS12ALDH1A1
SCHEMBL4353421 0.87 NOX4 (0.65) NOX4EGFRMAPTRGS12ALDH1A1
SCHEMBL4345390 0.87 MAPT (0.51) NOX4EGFRMAPTALDH1A1MEN1
SCHEMBL4357515 0.85 NOX4 (0.62) NOX4EGFRMAPTRGS12ALDH1A1
SCHEMBL4345601 0.84 MAPT (0.54) NOX4EGFRMAPTALDH1A1MEN1
SCHEMBL4346742 0.84 MAPT (0.45) NOX4EGFRMAPTMEN1KMT2A
SCHEMBL4345414 0.83 NOX4 (0.60) NOX4EGFRMAPTRGS12ALDH1A1
SCHEMBL4347478 0.82 NOX4 (0.59) NOX4EGFRMAPTRGS12ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2100876-A2 New compounds for the inhibition of rotamases and use thereof Jerini AG (DE) 2009-09-16 EP claimed
CN-1701061-A Novel compounds for inhibiting rotamase enzymes and uses thereof JERINI AG (DE) 2005-11-23 CN claimed
EP-1539683-A2 PHENOL DERIVATIVES AND THEIR USE AS ROTAMASE INHIBITORS Jerini AG (DE) 2005-06-15 EP claimed
WO-2004030664-A2 NEW COMPOUNDS FOR THE INHIBITION OF UNDESIRED CELL PROLIFERATION AND USE THEREOF JERINI AG (DE) 2004-04-15 WO claimed
WO-2004026815-A2 PHENOL DERIVATIVES AND THEIR USE AS ROTAMASE INHIBITORS JERINI AG (DE) 2004-04-01 WO claimed
EP-2100876-A2 New compounds for the inhibition of rotamases and use thereof Jerini AG (DE) 2009-09-16 EP disclosed