SCHEMBL4358462

SCHEMBL4358462

O=C(O)c1cc(NCc2ccccc2Sc2ccccc2)ccc1O

nearest known ligand 0.70

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
NOX4 Q9NPH5 3/20 0.70
EGFR P00533 10/20 0.59
RGS12 O14924 1/20 0.59
ALDH1A1 P00352 1/20 0.59
LCK P06239 1/20 0.59
MAPT P10636 1/20 0.59
CAMKK2 Q96RR4 1/20 0.59
TDP1 Q9NUW8 1/20 0.59
KDM4C Q9H3R0 3/20 0.56
PPARA Q07869 1/20 0.48
STING1 Q86WV6 1/20 0.48
SYK P43405 2/20 0.47
SMN1; SMN2 Q16637 1/20 0.45
HIF1A Q16665 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4357515 0.92 NOX4 (0.62) NOX4EGFRRGS12ALDH1A1LCK
SCHEMBL4345406 0.92 NOX4 (0.62) NOX4EGFRRGS12ALDH1A1LCK
SCHEMBL4355493 0.90 NOX4 (0.60) NOX4EGFRRGS12ALDH1A1LCK
SCHEMBL4345414 0.90 NOX4 (0.60) NOX4EGFRRGS12ALDH1A1LCK
SCHEMBL4347478 0.89 NOX4 (0.59) NOX4EGFRRGS12ALDH1A1LCK
SCHEMBL4341720 0.88 NOX4 (0.58) NOX4EGFRRGS12ALDH1A1LCK
SCHEMBL4346161 0.88 NOX4 (0.60) NOX4EGFRRGS12ALDH1A1LCK
SCHEMBL4353421 0.87 NOX4 (0.65) NOX4EGFRRGS12ALDH1A1LCK
SCHEMBL7803944 0.83 NOX4 (1.00) NOX4EGFRRGS12ALDH1A1LCK
SCHEMBL4343906 0.82 NOX4 (0.54) NOX4EGFRRGS12ALDH1A1LCK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2100876-A2 New compounds for the inhibition of rotamases and use thereof Jerini AG (DE) 2009-09-16 EP claimed
CN-1701061-A Novel compounds for inhibiting rotamase enzymes and uses thereof JERINI AG (DE) 2005-11-23 CN claimed
EP-1539683-A2 PHENOL DERIVATIVES AND THEIR USE AS ROTAMASE INHIBITORS Jerini AG (DE) 2005-06-15 EP claimed
WO-2004030664-A2 NEW COMPOUNDS FOR THE INHIBITION OF UNDESIRED CELL PROLIFERATION AND USE THEREOF JERINI AG (DE) 2004-04-15 WO claimed
WO-2004026815-A2 PHENOL DERIVATIVES AND THEIR USE AS ROTAMASE INHIBITORS JERINI AG (DE) 2004-04-01 WO claimed
EP-2100876-A2 New compounds for the inhibition of rotamases and use thereof Jerini AG (DE) 2009-09-16 EP disclosed