SCHEMBL4346879

SCHEMBL4346879

O=C(NCc1ccc(C(F)(F)F)cc1)Nc1ccc(O)c([N+](=O)[O-])c1

nearest known ligand 0.62

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
MTOR P42345 4/20 0.62
PRMT3 O60678 2/20 0.56
NAMPT P43490 4/20 0.56
ATG4B Q9Y4P1 1/20 0.53
GAA P10253 1/20 0.50
CA1 P00915 2/20 0.49
CA2 P00918 2/20 0.49
CA9 Q16790 2/20 0.49
CA12 O43570 1/20 0.49
CA7 P43166 1/20 0.48
MEN1 O00255 1/20 0.47
KMT2A Q03164 1/20 0.47
MCHR1 Q99705 1/20 0.47
TRPV1 Q8NER1 1/20 0.47
CNR1 P21554 1/20 0.45
ERCC1 P07992 1/20 0.44
ERCC4 Q92889 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4341575 0.88 MEN1 (0.59) MTORGAAMEN1KMT2A
SCHEMBL4347085 0.87 CA12 (0.61) MTORGAACA1CA2CA9
SCHEMBL4354177 0.84 MEN1 (0.57) PRMT3NAMPTATG4BGAACA1
SCHEMBL4347646 0.82 MTOR (0.70) MTORPRMT3NAMPTCA1CA2
SCHEMBL4348431 0.81 MTOR (0.68) MTORPRMT3NAMPTCA1CA2
SCHEMBL5906319 0.81 MTOR (0.59) MTORPRMT3NAMPTATG4BCA1
SCHEMBL4345484 0.78 HRAS (0.54) GAACA1CA2CA9CA12
SCHEMBL4341578 0.77 POLB (0.43) MTORATG4BCA1CA2CA12
SCHEMBL6672203 0.76 MEN1 (0.56) NAMPTCA1CA2CA9CA12
SCHEMBL26625460 0.76 MTOR (0.71) MTORPRMT3NAMPTMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-100546977-C Suppress the new compound and the application thereof of rotamase JERINI AG (DE) 2009-10-07 CN claimed
EP-2100876-A2 New compounds for the inhibition of rotamases and use thereof Jerini AG (DE) 2009-09-16 EP claimed
CN-1701061-A Novel compounds for inhibiting rotamase enzymes and uses thereof JERINI AG (DE) 2005-11-23 CN claimed
EP-2100876-A2 New compounds for the inhibition of rotamases and use thereof Jerini AG (DE) 2009-09-16 EP disclosed