SCHEMBL4347646

SCHEMBL4347646

O=C(NCc1ccc(C(F)(F)F)cc1)Nc1ccc(O)c(F)c1

nearest known ligand 0.70

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MTOR P42345 5/20 0.70
NAMPT P43490 3/20 0.62
PRMT3 O60678 1/20 0.61
TRPV1 Q8NER1 1/20 0.51
MCHR1 Q99705 1/20 0.51
CA1 P00915 1/20 0.50
CA2 P00918 1/20 0.50
CA7 P43166 1/20 0.50
CA9 Q16790 1/20 0.50
CNR1 P21554 1/20 0.49
ERCC1 P07992 1/20 0.49
ERCC4 Q92889 1/20 0.49
MEN1 O00255 1/20 0.49
KMT2A Q03164 1/20 0.49
EPHX2 P34913 1/20 0.49
LMNA P02545 1/20 0.48
SMN1; SMN2 Q16637 1/20 0.48
POLB P06746 1/20 0.48
RAB9A P51151 1/20 0.48
BAZ1A Q9NRL2 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4348348 0.87 MTOR (0.69) MTORNAMPTPRMT3TRPV1MCHR1
SCHEMBL21776629 0.87 RAB9A (0.63) MTORNAMPTPRMT3ERCC1ERCC4
SCHEMBL4348431 0.86 MTOR (0.68) MTORNAMPTPRMT3TRPV1MCHR1
SCHEMBL4354013 0.85 MEN1 (0.64) MTORMEN1KMT2ALMNASMN1; SMN2
SCHEMBL4357696 0.84 NAMPT (0.59) NAMPTCA1CA2CA9MEN1
SCHEMBL4346879 0.82 MTOR (0.62) MTORNAMPTPRMT3TRPV1MCHR1
SCHEMBL26625460 0.81 MTOR (0.71) MTORNAMPTPRMT3TRPV1MEN1
SCHEMBL28808075 0.78 MTOR (0.76) MTORNAMPTPRMT3CA1CA2
SCHEMBL4353993 0.78 MTOR (0.67) MTORNAMPTPRMT3TRPV1CA1
SCHEMBL4350068 0.78 MTOR (0.67) MTORNAMPTPRMT3TRPV1MCHR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-100546977-C Suppress the new compound and the application thereof of rotamase JERINI AG (DE) 2009-10-07 CN claimed
EP-2100876-A2 New compounds for the inhibition of rotamases and use thereof Jerini AG (DE) 2009-09-16 EP claimed
CN-1701061-A Novel compounds for inhibiting rotamase enzymes and uses thereof JERINI AG (DE) 2005-11-23 CN claimed
EP-2100876-A2 New compounds for the inhibition of rotamases and use thereof Jerini AG (DE) 2009-09-16 EP disclosed