SCHEMBL4348602

SCHEMBL4348602

CCCCCNC(=O)Nc1ccc(O)c(Cl)c1

nearest known ligand 0.74

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
EPHX2 P34913 6/20 0.74
EPHX1 P07099 10/20 0.65
MEN1 O00255 1/20 0.59
KMT2A Q03164 1/20 0.59
ALDH1A1 P00352 2/20 0.57
HTT P42858 1/20 0.57
CA1 P00915 1/20 0.54
CA2 P00918 1/20 0.54
MAPT P10636 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27761103 0.96 EPHX2 (0.67) EPHX2EPHX1MEN1KMT2AALDH1A1
SCHEMBL8777974 0.87 EPHX2 (0.80) EPHX2EPHX1MEN1KMT2AALDH1A1
SCHEMBL8391695 0.86 EPHX1 (0.67) EPHX2EPHX1ALDH1A1HTTMAPT
SCHEMBL13296457 0.84 EPHX2 (0.71) EPHX2EPHX1MEN1KMT2AALDH1A1
SCHEMBL4347034 0.84 EPHX2 (0.67) EPHX2EPHX1MEN1KMT2AALDH1A1
SCHEMBL8756365 0.83 EPHX2 (0.70) EPHX2EPHX1ALDH1A1HTTMAPT
SCHEMBL4346126 0.83 LMNA (0.61) EPHX2MEN1KMT2AALDH1A1HTT
SCHEMBL4343691 0.83 EPHX1 (0.60) EPHX2EPHX1MEN1KMT2AALDH1A1
SCHEMBL8602435 0.83 EPHX2 (0.69) EPHX2EPHX1MEN1KMT2AALDH1A1
SCHEMBL8602439 0.83 EPHX2 (0.69) EPHX2EPHX1MEN1KMT2AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2100876-A2 New compounds for the inhibition of rotamases and use thereof Jerini AG (DE) 2009-09-16 EP claimed
CN-1701061-A Novel compounds for inhibiting rotamase enzymes and uses thereof JERINI AG (DE) 2005-11-23 CN claimed
EP-2100876-A2 New compounds for the inhibition of rotamases and use thereof Jerini AG (DE) 2009-09-16 EP disclosed