SCHEMBL434875

SCHEMBL434875

O=C(NC(CN1CCCC1)c1ccccc1)C1(c2ccc3oc(=O)[nH]c3c2)CC1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TRPV1 Q8NER1 2/20 0.42
ROCK2 O75116 1/20 0.37
ROCK1 Q13464 1/20 0.37
GRIN2B Q13224 1/20 0.37
AURKA O14965 3/20 0.36
AURKB Q96GD4 2/20 0.36
CDC7 O00311 1/20 0.36
CHEK1 O14757 1/20 0.36
JAK2 O60674 1/20 0.36
PAK4 O96013 1/20 0.36
NTRK1 P04629 1/20 0.36
PRKCB P05771 1/20 0.36
INSR P06213 1/20 0.36
RET P07949 1/20 0.36
KIT P10721 1/20 0.36
FGFR1 P11362 1/20 0.36
PRKACA P17612 1/20 0.36
FLT4 P35916 1/20 0.36
KDR P35968 1/20 0.36
JAK3 P52333 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15385515 1.00 TRPV1 (0.42) TRPV1ROCK2ROCK1GRIN2BAURKA
SCHEMBL433021 0.91 TRPV1 (0.37) TRPV1ROCK2ROCK1GRIN2BKCNK3
SCHEMBL433022 0.91 TRPV1 (0.37) TRPV1ROCK2ROCK1GRIN2BKCNK3
SCHEMBL435712 0.90 TRPV1 (0.36) TRPV1ROCK2ROCK1GRIN2BAURKA
SCHEMBL435713 0.90 TRPV1 (0.36) TRPV1ROCK2ROCK1GRIN2BAURKA
SCHEMBL434161 0.89 TRPV1 (0.37) TRPV1ROCK2ROCK1AURKAAURKB
SCHEMBL434659 0.89 ROCK2 (0.45) ROCK2ROCK1
SCHEMBL434660 0.89 ROCK2 (0.45) ROCK2ROCK1
SCHEMBL434160 0.89 TRPV1 (0.37) TRPV1ROCK2ROCK1AURKAAURKB
SCHEMBL433872 0.89 MAOA (0.37) TRPV1ALDH1A1HTTRAB9ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012012410-A2 KAPPA OPIOID RECEPTOR AGONISTS DR. REDDY'S LABORATORIES LTD. (IN) 2012-01-26 WO disclosed