SCHEMBL4350107

SCHEMBL4350107

O=[N+]([O-])c1ccc(Sc2ccccc2CNc2ccc(O)c(F)c2)cc1

nearest known ligand 0.49

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ALDH3A1 P30838 1/20 0.49
MAOB P27338 1/20 0.44
ALDH1A1 P00352 3/20 0.44
MAPT P10636 3/20 0.44
MEN1 O00255 3/20 0.44
KMT2A Q03164 3/20 0.44
GAA P10253 2/20 0.41
PKM P14618 1/20 0.41
EGFR P00533 1/20 0.41
APP P05067 1/20 0.41
POLB P06746 1/20 0.40
KDM4E B2RXH2 1/20 0.40
RAB9A P51151 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
ALB P02768 1/20 0.40
PTPRF P10586 1/20 0.39
PTPN2 P17706 1/20 0.39
PTPN1 P18031 1/20 0.39
PTPN11 Q06124 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4347830 0.89 ALDH3A1 (0.46) ALDH3A1MAOBALDH1A1MAPTMEN1
SCHEMBL4343414 0.88 EGFR (0.56) ALDH3A1MAOBALDH1A1MAPTMEN1
SCHEMBL4342064 0.87 EGFR (0.44) ALDH3A1MAOBALDH1A1MAPTMEN1
SCHEMBL4342184 0.87 MAPT (0.47) MAOBALDH1A1MAPTMEN1KMT2A
SCHEMBL4349134 0.85 ALDH3A1 (0.47) ALDH3A1MAOBALDH1A1MAPTMEN1
SCHEMBL4341720 0.85 NOX4 (0.58) MAOBALDH1A1MAPTMEN1KMT2A
SCHEMBL4346787 0.85 NOX4 (0.45) ALDH3A1MAOBALDH1A1MAPTMEN1
SCHEMBL4358509 0.85 ALB (0.46) ALDH3A1MAOBALDH1A1MAPTMEN1
SCHEMBL4351067 0.85 MAPT (0.47) ALDH3A1ALDH1A1MAPTMEN1KMT2A
SCHEMBL4341774 0.83 MEN1 (0.50) ALDH3A1MAOBALDH1A1MAPTMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2100876-A2 New compounds for the inhibition of rotamases and use thereof Jerini AG (DE) 2009-09-16 EP claimed
CN-1701061-A Novel compounds for inhibiting rotamase enzymes and uses thereof JERINI AG (DE) 2005-11-23 CN claimed
EP-1539683-A2 PHENOL DERIVATIVES AND THEIR USE AS ROTAMASE INHIBITORS Jerini AG (DE) 2005-06-15 EP claimed
WO-2004030664-A2 NEW COMPOUNDS FOR THE INHIBITION OF UNDESIRED CELL PROLIFERATION AND USE THEREOF JERINI AG (DE) 2004-04-15 WO claimed
WO-2004026815-A2 PHENOL DERIVATIVES AND THEIR USE AS ROTAMASE INHIBITORS JERINI AG (DE) 2004-04-01 WO claimed
EP-2100876-A2 New compounds for the inhibition of rotamases and use thereof Jerini AG (DE) 2009-09-16 EP disclosed