SCHEMBL4350384

SCHEMBL4350384

Cc1cccnc1CN(Cc1ncccc1C)C1CCN(C(CC=O)N2CCOCC2)CC1

nearest known ligand 0.38

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ADAMTS4 O75173 1/20 0.38
MMP2 P08253 1/20 0.38
MMP9 P14780 1/20 0.38
MMP13 P45452 1/20 0.38
MMP14 P50281 1/20 0.38
ADAMTS5 Q9UNA0 1/20 0.38
CXCR4 P61073 3/20 0.36
EGLN1 Q9GZT9 1/20 0.36
IDH1 O75874 1/20 0.34
OPRL1 P41146 2/20 0.33
P2RX7 Q99572 5/20 0.33
ACKR3 P25106 1/20 0.31
CCR5 P51681 1/20 0.31
USP2 O75604 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5576989 0.81 CXCR4 (0.40) ADAMTS4MMP2MMP9MMP13MMP14
SCHEMBL2086000 0.76 CXCR4 (0.46) CXCR4ACKR3USP2
SCHEMBL23428555 0.74 KDM4E (0.46) CXCR4
SCHEMBL2084725 0.74 ALDH1A1 (0.42) CXCR4ACKR3USP2
SCHEMBL2081000 0.72 TDP1 (0.47) CXCR4ACKR3CCR5
SCHEMBL4535370 0.72 CCR5 (0.44) CXCR4ACKR3CCR5
SCHEMBL2083868 0.72 CXCR4 (0.42) ADAMTS4MMP2MMP9MMP13MMP14
SCHEMBL2082352 0.71 SMO (0.43) CXCR4ACKR3CCR5
SCHEMBL12935360 0.71 CCR5 (0.41) CXCR4ACKR3CCR5
SCHEMBL2083565 0.70 CXCR4 (0.37) CXCR4CCR5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1613613-A4 CXCR4 CHEMOKINE RECEPTOR BINDING COMPOUNDS ANORMED INC (CA) 2009-03-25 EP disclosed
EP-1613613-A2 CXCR4 CHEMOKINE RECEPTOR BINDING COMPOUNDS ANORMED INC. (CA) 2006-01-11 EP disclosed
WO-2004091518-A2 CXCR4 CHEMOKINE RECEPTOR BINDING COMPOUNDS ANORMED INC. (CA) 2004-10-28 WO disclosed