SCHEMBL4350893

SCHEMBL4350893

Cc1ccc(Sc2ccc([N+](=O)[O-])cc2CNc2ccc(O)c(Cl)c2)cc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALB P02768 1/20 0.46
TBXA2R P21731 1/20 0.45
PTGES O14684 1/20 0.44
MEN1 O00255 4/20 0.44
KMT2A Q03164 4/20 0.44
GAA P10253 3/20 0.44
MAPT P10636 3/20 0.44
ALDH1A1 P00352 2/20 0.44
RAB9A P51151 2/20 0.44
L3MBTL1 Q9Y468 1/20 0.44
APP P05067 1/20 0.44
CRHBP P24387 1/20 0.44
CASP3 P42574 1/20 0.44
CRHR2 Q13324 1/20 0.44
SENP8 Q96LD8 1/20 0.44
SENP7 Q9BQF6 1/20 0.44
SENP6 Q9GZR1 1/20 0.44
PDE7A Q13946 3/20 0.43
NPC1 O15118 2/20 0.41
PDE4B Q07343 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4345719 0.92 NPC1 (0.48) ALBMEN1KMT2AGAAMAPT
SCHEMBL4354093 0.90 TBXA2R (0.46) ALBTBXA2RPTGESMEN1KMT2A
SCHEMBL4341945 0.89 EGFR (0.53) ALBTBXA2RPTGESMEN1KMT2A
SCHEMBL4341695 0.88 ALB (0.48) ALBTBXA2RPTGESMEN1KMT2A
SCHEMBL4358509 0.88 ALB (0.46) ALBTBXA2RPTGESMEN1KMT2A
SCHEMBL4350329 0.86 PTGES (0.48) ALBTBXA2RPTGESMEN1KMT2A
SCHEMBL6225219 0.86 NPC1 (0.46) ALBTBXA2RPTGESMEN1KMT2A
SCHEMBL4342184 0.85 MAPT (0.47) ALBMEN1KMT2AGAAMAPT
SCHEMBL4344437 0.84 MAPT (0.48) TBXA2RPTGESMEN1KMT2AGAA
SCHEMBL4341835 0.84 TBXA2R (0.44) TBXA2RPTGESMEN1KMT2AGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2100876-A2 New compounds for the inhibition of rotamases and use thereof Jerini AG (DE) 2009-09-16 EP claimed
CN-1701061-A Novel compounds for inhibiting rotamase enzymes and uses thereof JERINI AG (DE) 2005-11-23 CN claimed
WO-2004030664-A2 NEW COMPOUNDS FOR THE INHIBITION OF UNDESIRED CELL PROLIFERATION AND USE THEREOF JERINI AG (DE) 2004-04-15 WO claimed
EP-2100876-A2 New compounds for the inhibition of rotamases and use thereof Jerini AG (DE) 2009-09-16 EP disclosed