SCHEMBL4350329

SCHEMBL4350329

Cc1ccc(Sc2ccc([N+](=O)[O-])cc2CNc2ccc(O)c(C(=O)O)c2)cc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGES O14684 1/20 0.48
ALDH1A1 P00352 3/20 0.47
MAPT P10636 3/20 0.47
NOX4 Q9NPH5 2/20 0.47
RGS12 O14924 1/20 0.47
EGFR P00533 1/20 0.47
LCK P06239 1/20 0.47
CAMKK2 Q96RR4 1/20 0.47
TDP1 Q9NUW8 1/20 0.47
LDHA P00338 1/20 0.46
LDHB P07195 1/20 0.46
HAO1 Q9UJM8 1/20 0.46
TBXA2R P21731 1/20 0.46
ALB P02768 1/20 0.45
KMT2A Q03164 4/20 0.45
MEN1 O00255 3/20 0.45
CRHBP P24387 1/20 0.45
CASP3 P42574 1/20 0.45
CRHR2 Q13324 1/20 0.45
SENP8 Q96LD8 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6225219 0.95 NPC1 (0.46) PTGESALDH1A1MAPTNOX4RGS12
SCHEMBL4347601 0.90 NPC1 (0.49) ALDH1A1MAPTNOX4RGS12EGFR
SCHEMBL4341945 0.87 EGFR (0.53) PTGESALDH1A1MAPTEGFRTDP1
SCHEMBL6225218 0.87 NPC1 (0.41) PTGESALDH1A1MAPTNOX4RGS12
SCHEMBL4350893 0.86 ALB (0.46) PTGESALDH1A1MAPTEGFRTBXA2R
SCHEMBL4341695 0.86 ALB (0.48) PTGESALDH1A1MAPTEGFRTDP1
SCHEMBL4358509 0.86 ALB (0.46) PTGESALDH1A1MAPTEGFRTBXA2R
SCHEMBL4341720 0.85 NOX4 (0.58) ALDH1A1MAPTNOX4RGS12EGFR
SCHEMBL4357515 0.83 NOX4 (0.62) ALDH1A1MAPTNOX4RGS12EGFR
SCHEMBL27749183 0.82 EGFR (0.67) ALDH1A1MAPTNOX4RGS12EGFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2100876-A2 New compounds for the inhibition of rotamases and use thereof Jerini AG (DE) 2009-09-16 EP claimed
CN-1701061-A Novel compounds for inhibiting rotamase enzymes and uses thereof JERINI AG (DE) 2005-11-23 CN claimed
WO-2004030664-A2 NEW COMPOUNDS FOR THE INHIBITION OF UNDESIRED CELL PROLIFERATION AND USE THEREOF JERINI AG (DE) 2004-04-15 WO claimed
EP-2100876-A2 New compounds for the inhibition of rotamases and use thereof Jerini AG (DE) 2009-09-16 EP disclosed