SCHEMBL435124

SCHEMBL435124

O=C(NCC(C1CCCCC1)N1CCCC1)C1(c2ccc3oc(=O)[nH]c3c2)CC1

nearest known ligand 0.36

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
TRPV1 Q8NER1 2/20 0.36
OPRD1 P41143 3/20 0.36
OPRM1 P35372 2/20 0.36
OPRK1 P41145 2/20 0.36
KCNH2 Q12809 2/20 0.35
MCHR2 Q969V1 1/20 0.35
MCHR1 Q99705 1/20 0.35
CYP3A4 P08684 3/20 0.33
CALCRL Q16602 3/20 0.33
ENPP2 Q13822 2/20 0.33
CYP2D6 P10635 1/20 0.33
TRPA1 O75762 4/20 0.33
PIK3CA P42336 1/20 0.33
CTSC P53634 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL434855 0.93 TRPA1 (0.38) TRPV1OPRD1OPRM1OPRK1KCNH2
SCHEMBL10084067 0.80 TRPV1 (0.41) TRPV1OPRD1OPRM1OPRK1KCNH2
SCHEMBL15380860 0.80 TRPV1 (0.41) TRPV1OPRD1OPRM1OPRK1KCNH2
SCHEMBL436051 0.78 KDM4E (0.36) TRPV1OPRK1CYP3A4CYP2D6
SCHEMBL10084062 0.77 MEN1 (0.44) TRPV1KCNH2MCHR2MCHR1CYP3A4
SCHEMBL434120 0.77 KCNH2 (0.37) TRPV1OPRD1OPRM1OPRK1KCNH2
SCHEMBL434121 0.77 KCNH2 (0.37) TRPV1OPRD1OPRM1OPRK1KCNH2
SCHEMBL432562 0.76 NOS3 (0.40) CYP3A4CYP2D6TRPA1
SCHEMBL15380879 0.74 TRPV1 (0.39) TRPV1OPRD1OPRM1OPRK1KCNH2
SCHEMBL434043 0.73 HTT (0.42) CYP3A4ENPP2CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012012410-A2 KAPPA OPIOID RECEPTOR AGONISTS DR. REDDY'S LABORATORIES LTD. (IN) 2012-01-26 WO claimed