SCHEMBL4351702

SCHEMBL4351702

CCOC(=O)CCNC(=O)Nc1cc(F)c(O)c(F)c1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.52
PTPN7 P35236 1/20 0.47
KDM4E B2RXH2 4/20 0.42
HSD17B10 Q99714 3/20 0.42
NPSR1 Q6W5P4 3/20 0.42
LMNA P02545 3/20 0.42
MAPK1 P28482 1/20 0.42
MEN1 O00255 3/20 0.42
KMT2A Q03164 3/20 0.42
MAPT P10636 5/20 0.41
HPGD P15428 3/20 0.41
HTT P42858 2/20 0.41
GAA P10253 2/20 0.40
SMN1; SMN2 Q16637 2/20 0.40
EPHX2 P34913 2/20 0.39
CASP3 P42574 1/20 0.38
TRPV1 Q8NER1 1/20 0.38
SENP7 Q9BQF6 1/20 0.38
NPC1 O15118 1/20 0.37
NLRP3 Q96P20 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4359582 0.86 ALDH1A1 (0.52) ALDH1A1PTPN7KDM4EHSD17B10NPSR1
SCHEMBL4345924 0.84 ALDH1A1 (0.52) ALDH1A1PTPN7KDM4EHSD17B10NPSR1
SCHEMBL4342431 0.84 ALDH1A1 (0.52) ALDH1A1PTPN7KDM4EHSD17B10NPSR1
SCHEMBL4358426 0.83 ALDH1A1 (0.43) ALDH1A1PTPN7KDM4EHSD17B10NPSR1
SCHEMBL4353970 0.81 ALDH1A1 (0.42) ALDH1A1PTPN7KDM4EHSD17B10NPSR1
SCHEMBL6226782 0.79 ALDH1A1 (0.50) ALDH1A1KDM4EHSD17B10NPSR1LMNA
SCHEMBL4346935 0.78 ALDH1A1 (0.49) ALDH1A1PTPN7KDM4EHSD17B10NPSR1
SCHEMBL6225668 0.78 ALDH1A1 (0.55) ALDH1A1PTPN7MAPTHTTEPHX2
SCHEMBL6228224 0.78 EPHX2 (0.47) ALDH1A1MEN1KMT2AMAPTHTT
SCHEMBL27519540 0.77 ALDH1A1 (0.82) ALDH1A1PTPN7KDM4EHSD17B10NPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2100876-A2 New compounds for the inhibition of rotamases and use thereof Jerini AG (DE) 2009-09-16 EP claimed
CN-1701061-A Novel compounds for inhibiting rotamase enzymes and uses thereof JERINI AG (DE) 2005-11-23 CN claimed
WO-2004030664-A2 NEW COMPOUNDS FOR THE INHIBITION OF UNDESIRED CELL PROLIFERATION AND USE THEREOF JERINI AG (DE) 2004-04-15 WO claimed
EP-2100876-A2 New compounds for the inhibition of rotamases and use thereof Jerini AG (DE) 2009-09-16 EP disclosed