SCHEMBL4359582

SCHEMBL4359582

CCOC(=O)CCNC(=O)Nc1ccc(O)c(F)c1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.52
PTPN7 P35236 1/20 0.52
KMT2A Q03164 4/20 0.48
MEN1 O00255 3/20 0.48
KDM4E B2RXH2 3/20 0.47
HSD17B10 Q99714 3/20 0.47
NPSR1 Q6W5P4 3/20 0.47
LMNA P02545 1/20 0.47
MAPK1 P28482 1/20 0.47
MAPT P10636 5/20 0.46
HPGD P15428 3/20 0.46
HTT P42858 2/20 0.46
SMN1; SMN2 Q16637 2/20 0.46
GAA P10253 2/20 0.44
RECQL P46063 1/20 0.42
EPHX2 P34913 2/20 0.42
POLB P06746 1/20 0.41
TDP1 Q9NUW8 1/20 0.41
CASP3 P42574 1/20 0.41
TRPV1 Q8NER1 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4351702 0.86 ALDH1A1 (0.52) ALDH1A1PTPN7KMT2AMEN1KDM4E
SCHEMBL4358300 0.85 ALDH1A1 (0.52) ALDH1A1PTPN7KMT2AMEN1KDM4E
SCHEMBL4346283 0.81 ALDH1A1 (0.49) ALDH1A1PTPN7KMT2AMEN1KDM4E
SCHEMBL27782774 0.80 RECQL (0.62) ALDH1A1KMT2AMEN1LMNAMAPT
SCHEMBL2270307 0.80 ESRRG (0.53) ALDH1A1KMT2AMEN1KDM4EMAPT
SCHEMBL4343691 0.79 EPHX1 (0.60) ALDH1A1KMT2AMEN1MAPTHTT
Hydrochloric Acid SCHEMBL322141 0.77 MEN1 (0.49) ALDH1A1KMT2AMEN1KDM4ELMNA
SCHEMBL27519540 0.77 ALDH1A1 (0.82) ALDH1A1PTPN7KMT2AMEN1KDM4E
SCHEMBL6670113 0.76 ALDH1A1 (0.51) ALDH1A1PTPN7KDM4EMAPTHTT
SCHEMBL6915485 0.76 ALDH1A1 (0.60) ALDH1A1PTPN7KMT2AMEN1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2100876-A2 New compounds for the inhibition of rotamases and use thereof Jerini AG (DE) 2009-09-16 EP claimed
CN-1701061-A Novel compounds for inhibiting rotamase enzymes and uses thereof JERINI AG (DE) 2005-11-23 CN claimed
EP-2100876-A2 New compounds for the inhibition of rotamases and use thereof Jerini AG (DE) 2009-09-16 EP disclosed