SCHEMBL4352185

SCHEMBL4352185

Cc1ccc(Sc2ccccc2CNc2ccc(O)c([N+](=O)[O-])c2)cc1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGFR P00533 1/20 0.55
MAPT P10636 8/20 0.46
ALDH1A1 P00352 5/20 0.46
L3MBTL1 Q9Y468 3/20 0.44
GAA P10253 2/20 0.44
MAPK1 P28482 2/20 0.44
KDM4E B2RXH2 1/20 0.44
ALDH3A1 P30838 1/20 0.44
PKM P14618 1/20 0.44
MEN1 O00255 3/20 0.43
KMT2A Q03164 3/20 0.43
LMNA P02545 2/20 0.43
NPSR1 Q6W5P4 2/20 0.43
ALOX12 P18054 1/20 0.43
HTT P42858 1/20 0.43
POLB P06746 1/20 0.42
ABCC1 P33527 1/20 0.40
ABCG2 Q9UNQ0 1/20 0.40
HPGD P15428 1/20 0.40
TDP1 Q9NUW8 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4350071 0.91 EGFR (0.59) EGFRMAPTALDH1A1L3MBTL1GAA
SCHEMBL4343414 0.90 EGFR (0.56) EGFRMAPTALDH1A1L3MBTL1GAA
SCHEMBL4351852 0.89 EGFR (0.55) EGFRMAPTALDH1A1L3MBTL1GAA
SCHEMBL4354926 0.89 EGFR (0.52) EGFRMAPTALDH1A1L3MBTL1GAA
SCHEMBL4353944 0.89 EGFR (0.52) EGFRMAPTALDH1A1L3MBTL1GAA
SCHEMBL4341945 0.88 EGFR (0.53) EGFRMAPTALDH1A1L3MBTL1GAA
SCHEMBL4341570 0.85 EGFR (0.53) EGFRMAPTALDH1A1L3MBTL1GAA
SCHEMBL4342105 0.85 ALDH3A1 (0.47) MAPTALDH1A1L3MBTL1GAAMAPK1
SCHEMBL4345796 0.83 EGFR (0.53) EGFRMAPTALDH1A1L3MBTL1GAA
SCHEMBL4358250 0.83 EGFR (0.57) EGFRMAPTALDH1A1L3MBTL1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2100876-A2 New compounds for the inhibition of rotamases and use thereof Jerini AG (DE) 2009-09-16 EP claimed
CN-1701061-A Novel compounds for inhibiting rotamase enzymes and uses thereof JERINI AG (DE) 2005-11-23 CN claimed
EP-1539683-A2 PHENOL DERIVATIVES AND THEIR USE AS ROTAMASE INHIBITORS Jerini AG (DE) 2005-06-15 EP claimed
WO-2004030664-A2 NEW COMPOUNDS FOR THE INHIBITION OF UNDESIRED CELL PROLIFERATION AND USE THEREOF JERINI AG (DE) 2004-04-15 WO claimed
WO-2004026815-A2 PHENOL DERIVATIVES AND THEIR USE AS ROTAMASE INHIBITORS JERINI AG (DE) 2004-04-01 WO claimed
EP-2100876-A2 New compounds for the inhibition of rotamases and use thereof Jerini AG (DE) 2009-09-16 EP disclosed