SCHEMBL4351852

SCHEMBL4351852

O=[N+]([O-])c1cc(NCc2ccccc2Sc2ccc(Cl)cc2)ccc1O

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGFR P00533 1/20 0.55
ALDH1A1 P00352 3/20 0.49
MAPT P10636 3/20 0.49
ALDH3A1 P30838 1/20 0.46
POLB P06746 2/20 0.45
PDE7A Q13946 3/20 0.44
PDE7B Q9NP56 2/20 0.44
GAA P10253 2/20 0.44
PKM P14618 1/20 0.44
BCL2L1 Q07817 2/20 0.42
PLA2G4A P47712 1/20 0.42
L3MBTL1 Q9Y468 2/20 0.42
KDM4E B2RXH2 1/20 0.42
MAPK1 P28482 1/20 0.42
IDO1 P14902 1/20 0.41
NPC1 O15118 2/20 0.40
SLC6A4 P31645 1/20 0.40
LMNA P02545 1/20 0.40
RAB9A P51151 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4350071 0.91 EGFR (0.59) EGFRALDH1A1MAPTALDH3A1PDE7A
SCHEMBL4343414 0.90 EGFR (0.56) EGFRALDH1A1MAPTALDH3A1GAA
SCHEMBL4345796 0.90 EGFR (0.53) EGFRALDH1A1MAPTALDH3A1POLB
SCHEMBL4341570 0.90 EGFR (0.53) EGFRALDH1A1MAPTALDH3A1POLB
SCHEMBL4352185 0.89 EGFR (0.55) EGFRALDH1A1MAPTALDH3A1POLB
SCHEMBL4351725 0.88 EGFR (0.53) EGFRALDH1A1MAPTPOLBPDE7A
SCHEMBL4358250 0.87 EGFR (0.57) EGFRALDH1A1MAPTALDH3A1POLB
SCHEMBL4354926 0.87 EGFR (0.52) EGFRALDH1A1MAPTALDH3A1PDE7A
SCHEMBL4353944 0.87 EGFR (0.52) EGFRALDH1A1MAPTALDH3A1POLB
SCHEMBL4345574 0.85 ALDH1A1 (0.49) EGFRALDH1A1MAPTALDH3A1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2100876-A2 New compounds for the inhibition of rotamases and use thereof Jerini AG (DE) 2009-09-16 EP claimed
CN-1701061-A Novel compounds for inhibiting rotamase enzymes and uses thereof JERINI AG (DE) 2005-11-23 CN claimed
EP-1539683-A2 PHENOL DERIVATIVES AND THEIR USE AS ROTAMASE INHIBITORS Jerini AG (DE) 2005-06-15 EP claimed
WO-2004030664-A2 NEW COMPOUNDS FOR THE INHIBITION OF UNDESIRED CELL PROLIFERATION AND USE THEREOF JERINI AG (DE) 2004-04-15 WO claimed
WO-2004026815-A2 PHENOL DERIVATIVES AND THEIR USE AS ROTAMASE INHIBITORS JERINI AG (DE) 2004-04-01 WO claimed
EP-2100876-A2 New compounds for the inhibition of rotamases and use thereof Jerini AG (DE) 2009-09-16 EP disclosed