SCHEMBL435254

SCHEMBL435254

Fc1ccc(C2CCCCC2)c(F)c1

nearest known ligand 0.59

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
OPRL1 P41146 9/20 0.59
PTGDR2 Q9Y5Y4 2/20 0.46
HTR2A P28223 1/20 0.43
HTR2C P28335 1/20 0.43
HTR2B P41595 1/20 0.43
NPC1 O15118 1/20 0.41
POLB P06746 1/20 0.41
RAB9A P51151 1/20 0.41
TP53 P04637 1/20 0.41
CHRNB2 P17787 1/20 0.40
CHRNB4 P30926 1/20 0.40
CHRNA3 P32297 1/20 0.40
CHRNA4 P43681 1/20 0.40
GRM2 Q14416 1/20 0.40
PTGDR Q13258 1/20 0.39
F2RL1 P55085 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL436724 0.98 OPRL1 (0.58) OPRL1PTGDR2HTR2AHTR2CHTR2B
SCHEMBL435077 0.94 OPRL1 (0.54) OPRL1PTGDR2HTR2AHTR2CHTR2B
SCHEMBL434354 0.89 OPRL1 (0.57) OPRL1HTR2AHTR2CHTR2BCHRNB2
SCHEMBL29266754 0.86 OPRL1 (0.56) OPRL1HTR2AHTR2CHTR2BTP53
SCHEMBL28095108 0.81 GAA (0.45) OPRL1PTGDR2NPC1RAB9A
SCHEMBL11773147 0.81 KDM1A (0.52) OPRL1PTGDR2NPC1CHRNB2CHRNB4
SCHEMBL24736536 0.80 OPRL1 (0.48) OPRL1PTGDR2HTR2AHTR2CHTR2B
SCHEMBL8785375 0.80 PTGDR2 (0.44) OPRL1PTGDR2CHRNB2CHRNB4CHRNA3
SCHEMBL5019341 0.80 OPRL1 (0.50) OPRL1HTR2AHTR2CHTR2BCHRNB2
SCHEMBL5100126 0.80 KDM1A (0.53) OPRL1PTGDR2NPC1RAB9APTGDR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109952300-B 5-or 8-substituted imidazo [1,5-a ] pyridines 百济神州有限公司 2022-01-18 CN disclosed
EP-2595985-A1 ISOXAZOLE, ISOTHIAZOLE, FURANE AND THIOPHENE COMPOUNDS AS MICROBICIDES Syngenta Participations AG (CH) 2013-05-29 EP disclosed
EP-2595984-A1 MICROBICIDES Syngenta Participations AG (CH) 2013-05-29 EP disclosed
WO-2012010567-A1 ISOXAZOLE, ISOTHIAZOLE, FURANE AND THIOPHENE COMPOUNDS AS MICROBICIDES SYNGENTA PARTICIPATIONS AG (CH) 2012-01-26 WO disclosed
WO-2012010568-A1 MICROBICIDES SYNGENTA PARTICIPATIONS AG (CH) 2012-01-26 WO disclosed