Bromide

Bromide

SCHEMBL4352867

Br.Br.CN(C)CCCN.c1ccc(P(c2ccccc2)c2ccccc2)cc1

nearest known ligand 0.46

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ACHEADRA1AADRA1BADRA1DADRA2AADRA2BADRA2CADRB1ADRB2ADRB3APH1AAPH1BCHRM2CHRM3EZH2GRIN2AHTR1AHTR1BHTR1DHTR1FHTR3ANCSTNP2RY12PSEN1PSEN2PSENENSIGMAR1SLC6A2SLC6A3SLC6A4

The experimentally established mechanism targets of Bromide. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
SIGMAR1 known ✓ Q99720 1/20 0.43
ADRA2C known ✓ P18825 1/20 0.37
TDP1 Q9NUW8 2/20 0.44
CYP3A4 P08684 1/20 0.44
HTR2A P28223 2/20 0.43
HRH1 P35367 2/20 0.43
TAAR1 Q96RJ0 1/20 0.39
CARM1 Q86X55 1/20 0.39
PRMT6 Q96LA8 1/20 0.39
PRMT8 Q9NR22 1/20 0.39
LSS P48449 1/20 0.39
ESR1 P03372 1/20 0.36
ESR2 Q92731 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10790182 0.82 CYP3A4 (0.60) TDP1CYP3A4HTR2AHRH1SIGMAR1
Bromide SCHEMBL4353499 0.81 CYP3A4 (0.44) TDP1CYP3A4HTR2AHRH1SIGMAR1
SCHEMBL28263824 0.80 CYP3A4 (0.63) TDP1CYP3A4HTR2AHRH1TAAR1
SCHEMBL9549618 0.79 CYP3A4 (0.46) TDP1CYP3A4HTR2AHRH1SIGMAR1
SCHEMBL6455349 0.79 CYP3A4 (0.46) TDP1CYP3A4HTR2AHRH1SIGMAR1
Bromide SCHEMBL9750017 0.79 SIGMAR1 (0.58) TDP1CYP3A4SIGMAR1TAAR1
SCHEMBL9549821 0.78 SIGMAR1 (0.47) TDP1CYP3A4HTR2AHRH1SIGMAR1
SCHEMBL9549513 0.78 SIGMAR1 (0.47) TDP1CYP3A4HTR2AHRH1SIGMAR1
Butylamine SCHEMBL28096832 0.76 CYP3A4 (0.52) TDP1CYP3A4HTR2AHRH1ESR1
Phenethylamine SCHEMBL29276774 0.76 SIGMAR1 (0.63) HTR2ASIGMAR1TAAR1CARM1PRMT6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009081417-A2 PROCESS FOR PREPARATION OF OLOPAT ADINE HYDROCHLORIDE INDOCO REMEDIES LIMITED (IN) 2009-07-02 WO disclosed