SCHEMBL4353864

SCHEMBL4353864

Oc1c(Br)cc(NC(=S)Nc2ccc(C(F)(F)F)cc2)cc1Br

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK1 P06493 1/20 0.51
MEN1 O00255 6/20 0.48
KMT2A Q03164 6/20 0.48
SMN1; SMN2 Q16637 5/20 0.48
MAPT P10636 5/20 0.48
LMNA P02545 3/20 0.48
HTT P42858 2/20 0.48
KDM4E B2RXH2 2/20 0.48
ALDH1A1 P00352 2/20 0.48
GAA P10253 1/20 0.48
KIF11 P52732 1/20 0.47
CA12 O43570 1/20 0.47
CA1 P00915 1/20 0.47
CA2 P00918 1/20 0.47
CA9 Q16790 1/20 0.47
EPHX2 P34913 1/20 0.46
HSPA9 P38646 1/20 0.44
MAPK1 P28482 1/20 0.44
NPSR1 Q6W5P4 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4348910 0.84 EPHX2 (0.69) MEN1KMT2ASMN1; SMN2MAPTHTT
SCHEMBL4351636 0.83 MEN1 (0.61) CDK1MEN1KMT2ASMN1; SMN2MAPT
SCHEMBL9453957 0.83 CDK1 (0.68) CDK1MEN1KMT2ASMN1; SMN2MAPT
SCHEMBL4358929 0.83 CDK1 (0.53) CDK1MEN1KMT2ASMN1; SMN2MAPT
SCHEMBL4359457 0.81 MAPT (0.57) CDK1MEN1KMT2ASMN1; SMN2MAPT
SCHEMBL18031170 0.80 GAA (0.69) CDK1MEN1KMT2ASMN1; SMN2MAPT
SCHEMBL4346604 0.79 MAPT (0.53) MEN1KMT2AMAPTHTTKDM4E
SCHEMBL4355354 0.78 ALDH1A1 (0.63) MEN1KMT2ASMN1; SMN2MAPTLMNA
SCHEMBL4348978 0.77 MEN1 (0.51) CDK1MEN1KMT2ASMN1; SMN2MAPT
SCHEMBL4349022 0.77 KMT2A (0.60) MEN1KMT2ASMN1; SMN2MAPTLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2100876-A2 New compounds for the inhibition of rotamases and use thereof Jerini AG (DE) 2009-09-16 EP claimed
CN-1701061-A Novel compounds for inhibiting rotamase enzymes and uses thereof JERINI AG (DE) 2005-11-23 CN claimed
EP-2100876-A2 New compounds for the inhibition of rotamases and use thereof Jerini AG (DE) 2009-09-16 EP disclosed