SCHEMBL4346604

SCHEMBL4346604

Oc1c(Br)cc(NC(=S)Nc2ccc(Cl)cc2)cc1Br

nearest known ligand 0.56

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
MAPT P10636 3/20 0.53
KDM4E B2RXH2 2/20 0.53
MAOB P27338 1/20 0.51
NOX1 Q9Y5S8 1/20 0.50
CNR1 P21554 2/20 0.49
NPC1 O15118 1/20 0.49
RAB9A P51151 1/20 0.49
ALDH1A1 P00352 3/20 0.49
GAA P10253 2/20 0.49
MMP2 P08253 1/20 0.48
EPHX1 P07099 1/20 0.47
THRB P10828 1/20 0.47
L3MBTL1 Q9Y468 1/20 0.47
CYP19A1 P11511 1/20 0.46
MEN1 O00255 1/20 0.46
HTT P42858 1/20 0.46
KMT2A Q03164 1/20 0.46
NPSR1 Q6W5P4 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4349866 0.86 IDO1 (0.56) MAPTMAOBALDH1A1MEN1HTT
SCHEMBL4355842 0.83 MEN1 (0.57) MAPTCNR1NPC1RAB9AALDH1A1
SCHEMBL4347956 0.82 ALDH1A1 (0.58) MAPTKDM4EMAOBNOX1CNR1
SCHEMBL4355354 0.82 ALDH1A1 (0.63) MAPTKDM4EMAOBNOX1NPC1
SCHEMBL5445907 0.81 MAPT (0.75) MAPTKDM4EMAOBNOX1CNR1
SCHEMBL8956455 0.81 MAPT (0.75) MAPTKDM4EMAOBNOX1CNR1
SCHEMBL11060530 0.80 CNR1 (0.70) MAPTKDM4EMAOBNOX1CNR1
SCHEMBL8956193 0.80 CNR1 (0.70) MAPTKDM4EMAOBNOX1CNR1
SCHEMBL4346164 0.79 MAOB (0.60) MAPTKDM4EMAOBNOX1NPC1
SCHEMBL4353864 0.79 CDK1 (0.51) MAPTKDM4EALDH1A1GAAL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2100876-A2 New compounds for the inhibition of rotamases and use thereof Jerini AG (DE) 2009-09-16 EP claimed
CN-1701061-A Novel compounds for inhibiting rotamase enzymes and uses thereof JERINI AG (DE) 2005-11-23 CN claimed
EP-2100876-A2 New compounds for the inhibition of rotamases and use thereof Jerini AG (DE) 2009-09-16 EP disclosed