SCHEMBL4353867

SCHEMBL4353867

Cc1cccc(C)c1NC(=O)Nc1cc(F)c(O)c(F)c1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.51
ALDH1A1 P00352 1/20 0.51
LMNA P02545 2/20 0.48
MAPT P10636 2/20 0.48
HTT P42858 2/20 0.48
ALOX15 P16050 1/20 0.48
RAB9A P51151 1/20 0.48
HSD17B10 Q99714 1/20 0.48
DDX3X O00571 1/20 0.46
POLB P06746 1/20 0.46
MEN1 O00255 1/20 0.46
NPC1 O15118 1/20 0.46
DRD2 P14416 1/20 0.45
HTR2A P28223 1/20 0.45
HTR2B P41595 1/20 0.45
IDH1 O75874 1/20 0.45
PKM P14618 1/20 0.44
EPHX1 P07099 1/20 0.43
NPY2R P49146 1/20 0.43
FPR2 P25090 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6228505 0.87 MAPT (0.54) KMT2AALDH1A1MAPTRAB9APOLB
SCHEMBL4353772 0.85 KMT2A (0.56) KMT2AALDH1A1LMNAMAPTHTT
SCHEMBL4354644 0.83 DDX3X (0.65) KMT2AALDH1A1MAPTHTTALOX15
SCHEMBL4353920 0.81 DHODH (0.60) KMT2AALDH1A1LMNAMAPTHTT
SCHEMBL4343772 0.81 KMT2A (0.55) KMT2AALDH1A1LMNAMAPTHTT
SCHEMBL4351694 0.81 CYP3A4 (0.47) KMT2AALDH1A1LMNAMAPTHTT
SCHEMBL30051979 0.79 MAPT (0.67) KMT2AALDH1A1LMNAMAPTHTT
SCHEMBL17438146 0.79 LMNA (0.66) KMT2AALDH1A1LMNAMAPTHTT
SCHEMBL4346830 0.79 LMNA (0.44) KMT2AALDH1A1LMNAMAPTHTT
SCHEMBL4350139 0.78 SMN1; SMN2 (0.63) KMT2AALDH1A1LMNAMAPTHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2100876-A2 New compounds for the inhibition of rotamases and use thereof Jerini AG (DE) 2009-09-16 EP claimed
CN-1701061-A Novel compounds for inhibiting rotamase enzymes and uses thereof JERINI AG (DE) 2005-11-23 CN claimed
EP-2100876-A2 New compounds for the inhibition of rotamases and use thereof Jerini AG (DE) 2009-09-16 EP disclosed