SCHEMBL4354067

SCHEMBL4354067

COc1cc(NC(=O)Nc2ccc(O)c(F)c2)cc(OC)c1OC

nearest known ligand 0.58

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
MAPT P10636 5/20 0.58
ALDH1A1 P00352 2/20 0.58
POLB P06746 2/20 0.58
GFER P55789 1/20 0.58
KMT2A Q03164 5/20 0.53
MEN1 O00255 4/20 0.53
RAB9A P51151 3/20 0.51
GAA P10253 1/20 0.51
SMN1; SMN2 Q16637 4/20 0.50
CYP3A4 P08684 1/20 0.49
CYP2C9 P11712 1/20 0.49
CYP2C19 P33261 1/20 0.49
NPC1 O15118 2/20 0.47
BCHE P06276 2/20 0.47
EPHX2 P34913 1/20 0.47
HTT P42858 1/20 0.46
ATM Q13315 1/20 0.45
HTR2A P28223 1/20 0.45
HTR2C P28335 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4348931 0.85 ALDH1A1 (0.56) MAPTALDH1A1POLBGFERKMT2A
SCHEMBL4341181 0.83 MAPT (0.58) MAPTALDH1A1POLBGFERKMT2A
SCHEMBL29663729 0.82 MAPT (0.69) MAPTALDH1A1POLBGFERKMT2A
SCHEMBL4354296 0.79 MEN1 (0.58) MAPTALDH1A1POLBGFERKMT2A
SCHEMBL4346922 0.78 TP53 (0.69) MAPTALDH1A1KMT2AMEN1RAB9A
SCHEMBL4347342 0.77 MEN1 (0.59) MAPTALDH1A1POLBGFERKMT2A
SCHEMBL6228505 0.77 MAPT (0.54) MAPTALDH1A1POLBGFERKMT2A
SCHEMBL4356336 0.76 KCNMA1 (0.59) MAPTALDH1A1POLBGFERKMT2A
SCHEMBL4347079 0.76 MAPT (0.49) MAPTALDH1A1POLBGFERKMT2A
SCHEMBL22279637 0.76 TNIK (0.52) MAPTALDH1A1POLBGFERKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-100546977-C Suppress the new compound and the application thereof of rotamase JERINI AG (DE) 2009-10-07 CN claimed
EP-2100876-A2 New compounds for the inhibition of rotamases and use thereof Jerini AG (DE) 2009-09-16 EP claimed
CN-1701061-A Novel compounds for inhibiting rotamase enzymes and uses thereof JERINI AG (DE) 2005-11-23 CN claimed
EP-2100876-A2 New compounds for the inhibition of rotamases and use thereof Jerini AG (DE) 2009-09-16 EP disclosed