SCHEMBL4354075

SCHEMBL4354075

CC(O)c1cc(NC(=S)Nc2cc(Cl)cc(Cl)c2)cc(Cl)c1O

nearest known ligand 0.47

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 1/20 0.46
MAOB P27338 2/20 0.45
ALDH1A1 P00352 5/20 0.45
MAPT P10636 5/20 0.45
MEN1 O00255 4/20 0.45
KMT2A Q03164 4/20 0.45
HPGD P15428 2/20 0.45
LMNA P02545 2/20 0.45
HTT P42858 2/20 0.44
XBP1 P17861 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
NPSR1 Q6W5P4 2/20 0.41
GAA P10253 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4355430 0.89 CNR1 (0.47) MAOBALDH1A1MAPTMEN1KMT2A
SCHEMBL4351932 0.88 KDM4E (0.41) IDO1MAOBALDH1A1MAPTMEN1
SCHEMBL4354098 0.86 ALDH1A1 (0.47) MAOBALDH1A1MAPTMEN1KMT2A
SCHEMBL4350857 0.84 ALDH1A1 (0.47) IDO1MAOBALDH1A1MAPTMEN1
SCHEMBL4349891 0.83 HTT (0.41) MAOBALDH1A1MAPTMEN1KMT2A
SCHEMBL4342470 0.82 IDO1 (0.60) IDO1MAOBALDH1A1MAPTMEN1
SCHEMBL4348451 0.80 PDE2A (0.48) MAOBALDH1A1MAPTMEN1KMT2A
SCHEMBL27782816 0.79 SMN1; SMN2 (0.52) ALDH1A1MAPTMEN1KMT2AHPGD
SCHEMBL4343912 0.78 HTT (0.47) MAOBALDH1A1MAPTMEN1KMT2A
SCHEMBL4347616 0.78 SMN1; SMN2 (0.57) ALDH1A1MAPTMEN1KMT2AHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2100876-A2 New compounds for the inhibition of rotamases and use thereof Jerini AG (DE) 2009-09-16 EP claimed
CN-1701061-A Novel compounds for inhibiting rotamase enzymes and uses thereof JERINI AG (DE) 2005-11-23 CN claimed
EP-2100876-A2 New compounds for the inhibition of rotamases and use thereof Jerini AG (DE) 2009-09-16 EP disclosed