SCHEMBL4354529

SCHEMBL4354529

CC(=O)Nc1ccc(Sc2ccccc2CNc2ccc(O)c(F)c2)cc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NOX4 Q9NPH5 2/20 0.41
MAOB P27338 1/20 0.41
EGFR P00533 1/20 0.41
HIF1A Q16665 1/20 0.40
SLC6A9 P48067 1/20 0.39
SMN1; SMN2 Q16637 4/20 0.39
MEN1 O00255 3/20 0.39
KMT2A Q03164 3/20 0.39
SLC6A2 P23975 1/20 0.39
SLC6A4 P31645 1/20 0.39
SLC6A3 Q01959 1/20 0.39
MAPK1 P28482 3/20 0.38
LMNA P02545 3/20 0.38
NPC1 O15118 2/20 0.38
ALOX15 P16050 1/20 0.38
CASP3 P42574 1/20 0.38
RAB9A P51151 1/20 0.38
SENP7 Q9BQF6 1/20 0.38
MAPT P10636 3/20 0.38
ALDH1A1 P00352 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4352975 0.90 GPR39 (0.41) MAOBHIF1ASLC6A9SMN1; SMN2MEN1
SCHEMBL4351072 0.87 NOX4 (0.41) NOX4EGFRHIF1ASLC6A9SMN1; SMN2
SCHEMBL4357506 0.87 EGFR (0.44) NOX4MAOBEGFRHIF1ASLC6A9
SCHEMBL4342291 0.86 MAPT (0.50) NOX4MAOBEGFRSMN1; SMN2MEN1
SCHEMBL4346787 0.86 NOX4 (0.45) NOX4MAOBEGFRHIF1ASMN1; SMN2
SCHEMBL4345414 0.86 NOX4 (0.60) NOX4EGFRHIF1ASLC6A9MEN1
SCHEMBL4341774 0.84 MEN1 (0.50) NOX4MAOBSMN1; SMN2MEN1KMT2A
SCHEMBL4359266 0.83 MEN1 (0.56) NOX4MAOBEGFRHIF1AMEN1
SCHEMBL4354926 0.83 EGFR (0.52) EGFRSMN1; SMN2MEN1KMT2AMAPK1
SCHEMBL4347664 0.83 SMN1; SMN2 (0.41) SLC6A9SMN1; SMN2MEN1KMT2ASLC6A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2100876-A2 New compounds for the inhibition of rotamases and use thereof Jerini AG (DE) 2009-09-16 EP claimed
CN-1701061-A Novel compounds for inhibiting rotamase enzymes and uses thereof JERINI AG (DE) 2005-11-23 CN claimed
EP-1539683-A2 PHENOL DERIVATIVES AND THEIR USE AS ROTAMASE INHIBITORS Jerini AG (DE) 2005-06-15 EP claimed
WO-2004026815-A2 PHENOL DERIVATIVES AND THEIR USE AS ROTAMASE INHIBITORS JERINI AG (DE) 2004-04-01 WO claimed
EP-2100876-A2 New compounds for the inhibition of rotamases and use thereof Jerini AG (DE) 2009-09-16 EP disclosed