SCHEMBL4355371

SCHEMBL4355371

O=C1[N]CN(c2ccccc2)C12CCNCC2

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD17B10 Q99714 4/20 0.57
TSHR P16473 4/20 0.42
USP2 O75604 5/20 0.41
CYP2D6 P10635 5/20 0.41
ALDH1A1 P00352 4/20 0.38
CYP3A4 P08684 3/20 0.38
CYP2C19 P33261 1/20 0.38
OPRM1 P35372 4/20 0.37
HTR3E A5X5Y0 1/20 0.37
HTR3B O95264 1/20 0.37
ADRB1 P08588 1/20 0.37
HTR3A P46098 1/20 0.37
HTR3D Q70Z44 1/20 0.37
HTR3C Q8WXA8 1/20 0.37
SIGMAR1 Q99720 1/20 0.37
OPRD1 P41143 3/20 0.36
OPRK1 P41145 3/20 0.36
OPRL1 P41146 3/20 0.36
TP53 P04637 3/20 0.36
CYP1A2 P05177 3/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4331085 0.73 HSD17B10 (0.59) HSD17B10TSHRUSP2CYP2D6ALDH1A1
SCHEMBL219618 0.73 HSD17B10 (1.00) HSD17B10OPRM1OPRD1OPRK1OPRL1
SCHEMBL7587764 0.73 HSD17B10 (1.00) HSD17B10OPRM1OPRD1OPRK1OPRL1
Ammonia Solution, Strong SCHEMBL1764035 0.72 HSD17B10 (0.97) HSD17B10OPRM1OPRD1OPRK1OPRL1
SCHEMBL20187016 0.72 HSD17B10 (0.57) HSD17B10TSHRUSP2CYP2D6OPRM1
SCHEMBL6162697 0.72 HSD17B10 (0.50) HSD17B10TSHRUSP2CYP2D6ALDH1A1
Hydrochloric Acid SCHEMBL6160546 0.72 HSD17B10 (0.97) HSD17B10OPRM1OPRD1OPRK1OPRL1
SCHEMBL3067132 0.71 OPRL1 (0.61) HSD17B10TSHRUSP2CYP2D6OPRM1
SCHEMBL4321885 0.70 HSD17B10 (0.55) HSD17B10TSHRUSP2CYP2D6ALDH1A1
Hydrochloric Acid SCHEMBL3231229 0.70 OPRL1 (0.60) HSD17B10TSHRUSP2CYP2D6OPRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1828227-A4 NEW PEPTIDIC AND PEPTIDOID BRADYKININ B1 RECEPTOR ANTAGONISTS AND USES THEREOF UNIV SHERBROOKE (CA) 2009-07-22 EP disclosed
EP-1828227-A1 NEW PEPTIDIC AND PEPTIDOID BRADYKININ B1 RECEPTOR ANTAGONISTS AND USES THEREOF Université de Sherbrooke (CA) 2007-09-05 EP disclosed
WO-2006017938-A1 NEW PEPTIDIC AND PEPTIDOID BRADYKININ B1 RECEPTOR ANTAGONISTS AND USES THEREOF UNIVERSITé DE SHERBROOKE (CA) 2006-02-23 WO disclosed