SCHEMBL4356401

SCHEMBL4356401

Oc1c(Br)cc(NCc2ccccc2Sc2ccccc2Cl)cc1Br

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACHE P22303 2/20 0.40
PRMT1 Q99873 1/20 0.40
CA1 P00915 1/20 0.40
ITGB2 P05107 1/20 0.39
ICAM1 P05362 1/20 0.39
ITGAL P20701 1/20 0.39
PRMT3 O60678 1/20 0.39
CARM1 Q86X55 1/20 0.39
PRMT6 Q96LA8 1/20 0.39
PRMT8 Q9NR22 1/20 0.39
MAOB P27338 1/20 0.38
MAPT P10636 3/20 0.38
GAA P10253 1/20 0.38
THRB P10828 1/20 0.38
ALDH1A1 P00352 2/20 0.38
CYP1A2 P05177 2/20 0.38
CYP2C9 P11712 2/20 0.38
CYP2C19 P33261 2/20 0.38
L3MBTL1 Q9Y468 2/20 0.38
HPGD P15428 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4347275 0.88 PRMT1 (0.42) ACHEPRMT1CA1ITGB2ICAM1
SCHEMBL4348016 0.85 MEN1 (0.41) ACHECA1MAOBMAPTALDH1A1
SCHEMBL4358682 0.85 SLC6A4 (0.46) ITGB2ICAM1ITGALMAOBMAPT
SCHEMBL4347048 0.84 CYP2C9 (0.47) PRMT1ITGB2ICAM1ITGALPRMT3
SCHEMBL4352803 0.84 SMN1; SMN2 (0.43) ACHEMAPTALDH1A1CYP2C9CYP2C19
SCHEMBL4351152 0.83 SLC6A4 (0.50) ACHECA1ITGB2ICAM1ITGAL
SCHEMBL6229046 0.80 CA1 (0.37) ACHEPRMT1CA1ITGB2ICAM1
SCHEMBL4348527 0.80 MAPT (0.46) ACHEPRMT1CA1ITGB2ICAM1
SCHEMBL4350338 0.80 MAPT (0.46) MAOBMAPTALDH1A1CYP2C9CYP2C19
SCHEMBL4344018 0.78 DHODH (0.38) ACHEPRMT1CA1ITGB2ICAM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2100876-A2 New compounds for the inhibition of rotamases and use thereof Jerini AG (DE) 2009-09-16 EP claimed
CN-1701061-A Novel compounds for inhibiting rotamase enzymes and uses thereof JERINI AG (DE) 2005-11-23 CN claimed
EP-1539683-A2 PHENOL DERIVATIVES AND THEIR USE AS ROTAMASE INHIBITORS Jerini AG (DE) 2005-06-15 EP claimed
WO-2004030664-A2 NEW COMPOUNDS FOR THE INHIBITION OF UNDESIRED CELL PROLIFERATION AND USE THEREOF JERINI AG (DE) 2004-04-15 WO claimed
WO-2004026815-A2 PHENOL DERIVATIVES AND THEIR USE AS ROTAMASE INHIBITORS JERINI AG (DE) 2004-04-01 WO claimed
EP-2100876-A2 New compounds for the inhibition of rotamases and use thereof Jerini AG (DE) 2009-09-16 EP disclosed