SCHEMBL4351152

SCHEMBL4351152

Oc1c(Br)cc(NCc2ccccc2Sc2cccc(Cl)c2)cc1Br

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A4 P31645 2/20 0.50
SLC6A2 P23975 1/20 0.50
SLC6A3 Q01959 1/20 0.50
SMN1; SMN2 Q16637 1/20 0.41
ALDH1A1 P00352 2/20 0.37
CYP2C9 P11712 2/20 0.37
CYP2C19 P33261 2/20 0.37
CYP1A2 P05177 1/20 0.37
HPGD P15428 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
RHEB Q15382 1/20 0.37
MAOB P27338 1/20 0.36
SLC6A9 P48067 3/20 0.35
ACHE P22303 2/20 0.35
CA2 P00918 1/20 0.35
MEN1 O00255 3/20 0.34
KMT2A Q03164 3/20 0.34
MAPT P10636 2/20 0.34
POLB P06746 1/20 0.34
PLEC Q15149 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4354940 0.88 SLC6A4 (0.52) SLC6A4SLC6A2SLC6A3SMN1; SMN2ALDH1A1
SCHEMBL4358682 0.88 SLC6A4 (0.46) SLC6A4SLC6A2SLC6A3SMN1; SMN2ALDH1A1
SCHEMBL4352803 0.87 SMN1; SMN2 (0.43) SLC6A4SLC6A2SLC6A3SMN1; SMN2ALDH1A1
SCHEMBL4351653 0.86 SLC6A4 (0.53) SLC6A4SLC6A2SLC6A3SMN1; SMN2ALDH1A1
SCHEMBL4348016 0.86 MEN1 (0.41) SLC6A4SLC6A2SLC6A3SMN1; SMN2ALDH1A1
SCHEMBL12846505 0.84 SLC6A4 (0.51) SLC6A4SLC6A2SLC6A3SMN1; SMN2ALDH1A1
SCHEMBL4356401 0.83 ACHE (0.40) SMN1; SMN2ALDH1A1CYP2C9CYP2C19CYP1A2
SCHEMBL6230536 0.81 SLC6A4 (0.46) SLC6A4SLC6A2SLC6A3SMN1; SMN2ALDH1A1
SCHEMBL4345562 0.81 SLC6A2 (0.50) SLC6A4SLC6A2SLC6A3SMN1; SMN2ALDH1A1
SCHEMBL4350338 0.81 MAPT (0.46) SLC6A4SLC6A2SLC6A3SMN1; SMN2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2100876-A2 New compounds for the inhibition of rotamases and use thereof Jerini AG (DE) 2009-09-16 EP claimed
CN-1701061-A Novel compounds for inhibiting rotamase enzymes and uses thereof JERINI AG (DE) 2005-11-23 CN claimed
EP-1539683-A2 PHENOL DERIVATIVES AND THEIR USE AS ROTAMASE INHIBITORS Jerini AG (DE) 2005-06-15 EP claimed
WO-2004030664-A2 NEW COMPOUNDS FOR THE INHIBITION OF UNDESIRED CELL PROLIFERATION AND USE THEREOF JERINI AG (DE) 2004-04-15 WO claimed
WO-2004026815-A2 PHENOL DERIVATIVES AND THEIR USE AS ROTAMASE INHIBITORS JERINI AG (DE) 2004-04-01 WO claimed
EP-2100876-A2 New compounds for the inhibition of rotamases and use thereof Jerini AG (DE) 2009-09-16 EP disclosed