SCHEMBL4358682

SCHEMBL4358682

Oc1c(Br)cc(NCc2ccccc2Sc2ccc(Cl)cc2)cc1Br

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A4 P31645 3/20 0.46
MEN1 O00255 4/20 0.40
KMT2A Q03164 4/20 0.40
ALDH1A1 P00352 3/20 0.40
LMNA P02545 2/20 0.40
BLM P54132 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40
NOD2 Q9HC29 1/20 0.40
CYP2C9 P11712 3/20 0.39
CYP2C19 P33261 2/20 0.39
CYP1A2 P05177 2/20 0.39
HPGD P15428 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
HDAC1 Q13547 1/20 0.38
HDAC8 Q9BY41 1/20 0.38
HDAC6 Q9UBN7 1/20 0.38
POLB P06746 4/20 0.38
SLC6A2 P23975 2/20 0.38
SLC6A3 Q01959 2/20 0.38
SMN1; SMN2 Q16637 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4352803 0.90 SMN1; SMN2 (0.43) SLC6A4MEN1KMT2AALDH1A1LMNA
SCHEMBL4351152 0.88 SLC6A4 (0.50) SLC6A4MEN1KMT2AALDH1A1NPSR1
SCHEMBL4348016 0.88 MEN1 (0.41) SLC6A4MEN1KMT2AALDH1A1LMNA
SCHEMBL4350338 0.88 MAPT (0.46) SLC6A4MEN1KMT2AALDH1A1LMNA
SCHEMBL4349840 0.87 SLC6A4 (0.48) SLC6A4MEN1KMT2AALDH1A1LMNA
SCHEMBL4347073 0.85 MEN1 (0.49) SLC6A4MEN1KMT2AALDH1A1LMNA
SCHEMBL4356401 0.85 ACHE (0.40) MEN1KMT2AALDH1A1CYP2C9CYP2C19
SCHEMBL4346948 0.84 MEN1 (0.42) SLC6A4MEN1KMT2AALDH1A1LMNA
SCHEMBL4353810 0.84 MEN1 (0.58) SLC6A4MEN1KMT2AALDH1A1LMNA
SCHEMBL4349811 0.82 MAOB (0.41) MEN1KMT2AALDH1A1LMNACYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2100876-A2 New compounds for the inhibition of rotamases and use thereof Jerini AG (DE) 2009-09-16 EP claimed
CN-1701061-A Novel compounds for inhibiting rotamase enzymes and uses thereof JERINI AG (DE) 2005-11-23 CN claimed
EP-1539683-A2 PHENOL DERIVATIVES AND THEIR USE AS ROTAMASE INHIBITORS Jerini AG (DE) 2005-06-15 EP claimed
WO-2004030664-A2 NEW COMPOUNDS FOR THE INHIBITION OF UNDESIRED CELL PROLIFERATION AND USE THEREOF JERINI AG (DE) 2004-04-15 WO claimed
WO-2004026815-A2 PHENOL DERIVATIVES AND THEIR USE AS ROTAMASE INHIBITORS JERINI AG (DE) 2004-04-01 WO claimed
EP-2100876-A2 New compounds for the inhibition of rotamases and use thereof Jerini AG (DE) 2009-09-16 EP disclosed